Target Details
| UniProt AC | O96020 |
|---|---|
| Gene Symbol | CCNE2 |
| Protein Name | G1/S-specific cyclin-E2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) |
Summary
- Multi-target molecules 504
- Clinical molecules 252
- Avg pChEMBL 7.06
KEGG Pathways (17)
- Cell cycle
- Cellular senescence
- Cushing syndrome
- Epstein-Barr virus infection
- Gastric cancer
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Measles
- MicroRNAs in cancer
- Oocyte meiosis
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (504)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GXAMBYHREJMOKQ
|
9.0 | IC50 | 11 | Yes | |
PIMQWRZWLQKKBJ
|
9.0 | Ki | 36 | — | |
TVARIYLSKVWCHN
|
9.0 | Ki | 11 | — | |
CGJRRFJDMMUHJW
|
8.7 | IC50 | 5 | Yes | |
DUEBWXVTFJJWCJ
|
8.7 | IC50 | 11 | Yes | |
DYTKVFHLKPDNRW
|
8.7 | Ki | 23 | Yes | |
ISZYBQYCHOZPBF
|
8.7 | IC50 | 11 | Yes | |
NOCXREGHIRXAHY
|
8.7 | IC50 | 3 | — | |
VAOAJUWPEYBTAB
|
8.7 | IC50 | 9 | Yes | |
ZJDFSKSBQBPOSK
|
8.7 | IC50 | 24 | Yes | |
AEKRDXUBYIUNBW
|
8.5 | IC50 | 3 | — | |
FDWQSLRDIBRKEI
|
8.5 | IC50 | 9 | Yes | |
GAIOPWBQKZMUNO
|
8.5 | Ki | 13 | — | |
GQTPCOMZBGFWLQ
|
8.5 | IC50 | 11 | Yes | |
MPJITOINOMJIJI
|
8.5 | IC50 | 11 | Yes | |
RAKYKJWUUUKCCW
|
8.5 | IC50 | 3 | — | |
RETDFEDFSXGWJW
|
8.5 | IC50 | 3 | — | |
XERLASHNAPKEEL
|
8.5 | IC50 | 7 | Yes | |
XLSYZSRXVVCHLS
|
8.5 | IC50 | 48 | — | |
AWZLLTSFYOFJHT
|
8.4 | IC50 | 3 | — | |
IHQAQVKWEYAOFQ
|
8.4 | IC50 | 5 | Yes | |
KAJOBXDSMROSCM
|
8.4 | IC50 | 3 | — | |
LOQNAQWIGMNXII
|
8.4 | IC50 | 9 | Yes | |
QMIDZOGAPGBZSC
|
8.4 | IC50 | 4 | — | |
SFGWUTHNZVSATD
|
8.4 | IC50 | 11 | Yes | |
VVEJXZWNRXJDBL
|
8.4 | IC50 | 3 | — | |
ZSPQUICTVOBVJJ
|
8.4 | IC50 | 4 | — | |
QIEKHLDZKRQLLN
|
8.3 | IC50 | 9 | — | |
AEKRDXUBYIUNBW
|
8.3 | IC50 | 3 | — | |
AWZLLTSFYOFJHT
|
8.3 | IC50 | 3 | — | |
DLPIYBKBHMZCJI
|
8.3 | Ki | 11 | — | |
FETXAWXOSWHGHF
|
8.3 | IC50 | 9 | Yes | |
GFXMFSCCEVADLF
|
8.3 | IC50 | 11 | Yes | |
HFMGTBLBSYZDFW
|
8.3 | IC50 | 8 | Yes | |
LBXKLCPOKBPOST
|
8.3 | IC50 | 5 | Yes | |
NDUNPMAPBHPTHE
|
8.3 | IC50 | 8 | Yes | |
VBDQMJNIWDFAKI
|
8.3 | IC50 | 8 | Yes | |
FIZSPBCJAWUURL
|
8.2 | IC50 | 3 | — | |
HCSOUJXRCJMNFB
|
8.2 | IC50 | 8 | Yes | |
OIINJADYHQPDPP
|
8.2 | IC50 | 4 | — | |
PHEMXOLLNFYYLK
|
8.2 | IC50 | 8 | Yes | |
BUVUGYVWVBFUMI
|
8.2 | Ki | 11 | — | |
RRLAXKDDEVSLJO
|
8.2 | IC50 | 5 | Yes | |
SXMLFYVKHGTDIW
|
8.2 | IC50 | 5 | Yes | |
UYNSEUPNWDBKBJ
|
8.2 | IC50 | 3 | — | |
AYJNSWHEIFEJGX
|
8.1 | IC50 | 5 | Yes | |
BGZVCNSRUXWDPB
|
8.1 | IC50 | 5 | Yes | |
CGKJOISVQXEPSG
|
8.1 | Ki | 9 | — | |
WKTFLAJOGAQWFX
|
8.1 | IC50 | 5 | Yes | |
ZSPQUICTVOBVJJ
|
8.1 | IC50 | 3 | — |