Target Details
| UniProt AC | O96013 |
|---|---|
| Gene Symbol | PAK4 |
| Protein Name | Serine/threonine-protein kinase PAK 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00786 (PBD) PF00069 (Pkinase) |
Summary
- Multi-target molecules 189
- Clinical molecules 15
- Avg pChEMBL 6.84
KEGG Pathways (10)
Active Molecules (189)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VWACUNWBMWWMPJ
|
6.2 | Ki | 18 | — | |
XXSPHNFKLDJDAK
|
6.2 | Ki | 26 | — | |
ZLLCVOJWNDZXIO
|
6.2 | Ki | 11 | — | |
ZVWRFVCNQOECJS
|
6.2 | Ki | 71 | — | |
FQPRRMPEEHYYNP
|
6.2 | IC50 | 2 | — | |
UDFJBAMCRJJGMV
|
6.2 | IC50 | 2 | — | |
UHEFRVBGJORHNV
|
6.2 | IC50 | 4 | — | |
ZBNZXTGUTAYRHI
|
6.1 | Kd | 102 | Yes | |
AEYLJTAIDDIOBA
|
6.1 | Ki | 53 | — | |
CYLGCMABIBXHIQ
|
6.1 | Ki | 16 | — | |
HZPACYSNLOCDLW
|
6.1 | Ki | 48 | — | |
KAZJIBCOYQRDGG
|
6.1 | Ki | 16 | — | |
MASJMHFQMYAPJR
|
6.1 | Ki | 41 | — | |
OLUKILHGKRVDCT
|
6.1 | Ki | 44 | Yes | |
UGUZOLHBLLTLBA
|
6.1 | Ki | 15 | — | |
UZFPGFONVYFSRR
|
6.1 | Ki | 16 | — | |
ZGDYBJXDIXVTLV
|
6.1 | Ki | 54 | — | |
OFBJDUJZLIENIO
|
6.1 | Ki | 2 | — | |
HUXYBQXJVXOMKX
|
6.1 | Kd | 28 | — | |
YOVVNQKCSKSHKT
|
6.0 | Kd | 15 | — | |
CYXJGDDHTZEOTA
|
6.0 | Ki | 2 | — | |
MVIXSPFFCUNNHO
|
6.0 | IC50 | 2 | — | |
WZQNDAXWFUAUMW
|
6.0 | Ki | 2 | — | |
BPNUQXPIQBZCMR
|
6.0 | Kd | 83 | Yes | |
ACSYKUPGCXYRRO
|
6.0 | Ki | 26 | — | |
AUDNGNGLLRZLDR
|
6.0 | Ki | 33 | — | |
DPEXRCOBPACFOO
|
6.0 | Ki | 36 | — | |
DYNHJHQFHQTFTP
|
6.0 | Kd | 38 | — | |
GHPFQRTVUDXWCC
|
6.0 | Ki | 35 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MFAQYJIYDMLAIM
|
6.0 | Kd | 130 | Yes | |
NKGLJTITEFZKAN
|
6.0 | Ki | 35 | — | |
OTVCFDOYUHREFJ
|
6.0 | Ki | 26 | — | |
QLWUDWMYFSWGHK
|
6.0 | Ki | 22 | — | |
SBFPHSVZEXSHTL
|
6.0 | Ki | 62 | — | |
WZISGNDZZPSYRP
|
6.0 | Ki | 20 | — | |
ZDPGLLQANLROFM
|
6.0 | Ki | 17 | — |