Target Details
| UniProt AC | O96013 |
|---|---|
| Gene Symbol | PAK4 |
| Protein Name | Serine/threonine-protein kinase PAK 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00786 (PBD) PF00069 (Pkinase) |
Summary
- Multi-target molecules 189
- Clinical molecules 15
- Avg pChEMBL 6.84
KEGG Pathways (10)
Active Molecules (189)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LDWBULFGVRAVMR
|
6.6 | Ki | 3 | — | |
BWMYPJVJYVLPIC
|
6.6 | IC50 | 2 | — | |
GDXPJJSKIKGEOQ
|
6.5 | Ki | 2 | — | |
GIWIOFZXFSKQTE
|
6.5 | IC50 | 4 | — | |
ADMFLILDQJSEIK
|
6.5 | Ki | 72 | — | |
JNXJKTXDSPWNRP
|
6.5 | Ki | 30 | — | |
UDFDIIVNIYWXDM
|
6.5 | Ki | 74 | — | |
UYGYYOIUVFMGKQ
|
6.5 | Ki | 30 | — | |
KOZFSFOOLUUIGY
|
6.5 | Kd | 88 | Yes | |
OEHGEOWDIWFUCT
|
6.5 | IC50 | 2 | — | |
ZDSMRCALKWRRFK
|
6.5 | Ki | 2 | — | |
LJIAMQXFSCERQG
|
6.4 | Ki | 2 | — | |
ZNXHSLJBVPFPJV
|
6.4 | IC50 | 2 | — | |
BLQYVHBZHAISJM
|
6.4 | Ki | 54 | — | |
CTKWGPSDOQLVKK
|
6.4 | IC50 | 2 | — | |
QQWUGDVOUVUTOY
|
6.4 | Ki | 231 | Yes | |
RGOPHVZLEMGMBZ
|
6.4 | Ki | 20 | — | |
UMTWTCVTRDYHQQ
|
6.4 | Ki | 56 | — | |
DYLHVDVCWIEYSA
|
6.3 | Ki | 2 | — | |
ORWIYCURPDKSBI
|
6.3 | IC50 | 15 | Yes | |
PNUWZKCIGDXYNR
|
6.3 | IC50 | 2 | — | |
ATGVCJYHNOSZEV
|
6.3 | Ki | 23 | — | |
FTKWFHKMPQIDLM
|
6.3 | Ki | 5 | — | |
GRXRHIRKSUPJKF
|
6.3 | Ki | 2 | — | |
NOBMKUVHFRVBES
|
6.3 | Ki | 19 | — | |
RFBPWKMQWSIPEO
|
6.3 | Ki | 28 | — | |
SACRIVBWIXWZAH
|
6.3 | Ki | 4 | — | |
YEHCNYAQEBQCCS
|
6.3 | Ki | 74 | — | |
ZGZVRPRSFXRGCF
|
6.3 | Ki | 76 | — | |
ZMNWFTYYYCSSTF
|
6.3 | Ki | 18 | — | |
DKZYXHCYPUVGAF
|
6.3 | Kd | 112 | — | |
IXAOAKWGJQGTSH
|
6.3 | IC50 | 3 | — | |
WNBOTPDRPIQGEY
|
6.3 | IC50 | 2 | — | |
FQADRNAKESOLCX
|
6.3 | IC50 | 2 | — | |
LXAVLHJMLKIDME
|
6.3 | Ki | 3 | — | |
UIBDEIGYCMBVOR
|
6.3 | IC50 | 2 | — | |
LBCUDZVMIGSKCJ
|
6.2 | Ki | 2 | — | |
WINHZLLDWRZWRT
|
6.2 | IC50 | 201 | Yes | |
DEQUZSQDCDHROJ
|
6.2 | IC50 | 2 | — | |
FHIUVWSTDWOTLV
|
6.2 | Ki | 2 | — | |
SIXQNSLYMZXLPF
|
6.2 | Ki | 3 | — | |
XCEVZNDXUCATCI
|
6.2 | Ki | 2 | — | |
XQFLBDFFGHEFGF
|
6.2 | Ki | 2 | — | |
AQKQATGZIKRZMQ
|
6.2 | Ki | 16 | — | |
GDYZFFBMSBDTAA
|
6.2 | Ki | 60 | — | |
GIAAJPPEMQIXPQ
|
6.2 | Ki | 3 | — | |
IFPPYSWJNWHOLQ
|
6.2 | Ki | 52 | Yes | |
NVRXTLZYXZNATH
|
6.2 | Ki | 47 | Yes | |
PCQMERRARZKTPW
|
6.2 | Ki | 68 | — | |
VSVWQTDDGQSGHP
|
6.2 | Ki | 51 | — |