Target Details
| UniProt AC | O96013 |
|---|---|
| Gene Symbol | PAK4 |
| Protein Name | Serine/threonine-protein kinase PAK 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00786 (PBD) PF00069 (Pkinase) |
Summary
- Multi-target molecules 189
- Clinical molecules 15
- Avg pChEMBL 6.84
KEGG Pathways (10)
Active Molecules (189)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PROLIXHVRCJEFH
|
7.3 | Ki | 46 | — | |
TVUWQDLBEOZVOU
|
7.3 | Ki | 41 | — | |
VXYDJXMHISGSDA
|
7.3 | Ki | 59 | — | |
XUFLBSMTYMFOQH
|
7.3 | Ki | 43 | — | |
YFNWWNRZJGMDBR
|
7.3 | Kd | 35 | — | |
JJGSOVIZOMZMCS
|
7.2 | Ki | 35 | — | |
VWVYILCFSYNJHF
|
7.2 | Ki | 49 | — | |
ASLFQIAAFMLPFR
|
7.2 | Ki | 3 | — | |
MJHOMTRKVMKCNE
|
7.1 | IC50 | 12 | — | |
XVBWTZHNQZHFHR
|
7.1 | Ki | 5 | — | |
CHTMRWQLNNRRFJ
|
7.1 | Ki | 70 | — | |
CKGISEYYRLOYIJ
|
7.1 | Ki | 2 | — | |
KTWBYGUSEYSRND
|
7.1 | Ki | 28 | — | |
SMRWVXLSRJWVBF
|
7.1 | Ki | 25 | — | |
SRONQUHCRFZABC
|
7.1 | Ki | 28 | — | |
UOVCGJXDGOGOCZ
|
7.1 | Ki | 59 | — | |
WJHAMZUWDONFQH
|
7.0 | IC50 | 2 | — | |
AONLJIQJHRPQBZ
|
7.0 | Ki | 2 | — | |
MRFOPLWJZULAQD
|
7.0 | IC50 | 2 | — | |
OUJZYQBEFNDJQN
|
7.0 | Ki | 71 | — | |
PLHUMPJXRHMFFR
|
7.0 | Ki | 28 | — | |
RWKDVIAVTRRJIR
|
7.0 | Ki | 23 | — | |
RYYNGWLOYLRZLK
|
7.0 | Ki | 104 | — | |
VVEGARMQKNYDID
|
7.0 | Ki | 24 | — | |
XPHWIERLJBFPFV
|
7.0 | Ki | 69 | — | |
DXUVJKCCXSAUKZ
|
7.0 | Ki | 2 | — | |
DGLFSNZWRYADFC
|
7.0 | IC50 | 12 | — | |
LOLPPWBBNUVNQZ
|
7.0 | Kd | 97 | Yes | |
NHHQJBCNYHBUSI
|
7.0 | Kd | 220 | — | |
CNQGNADBGYCKKV
|
6.9 | Ki | 25 | — | |
HOYRWTWZUFFACV
|
6.9 | Ki | 28 | — | |
LCHCSKHPVCDXAU
|
6.9 | Ki | 30 | — | |
PMXCMJLOPOFPBT
|
6.9 | IC50 | 17 | Yes | |
TUBXJQSNTKADJB
|
6.9 | IC50 | 5 | — | |
MERRGQWRCCBKDB
|
6.8 | Ki | 2 | — | |
CHADTINFLWZSKR
|
6.8 | Ki | 26 | — | |
RGNHKJWHFIPHIM
|
6.8 | Ki | 66 | — | |
SKKRZILJUKYLJS
|
6.8 | Ki | 25 | — | |
XZONYYFHQICDAM
|
6.8 | Ki | 19 | — | |
ZWVZORIKUNOTCS
|
6.8 | Ki | 69 | — | |
DUBHPLWTLUVGNU
|
6.8 | IC50 | 5 | — | |
HHJSKDRCUMVWKF
|
6.8 | IC50 | 7 | — | |
IAYGCINLNONXHY
|
6.8 | Kd | 50 | — | |
FPENQVXQIUJGIO
|
6.8 | IC50 | 2 | — | |
FDVSOQRNTAPCHB
|
6.7 | Ki | 40 | — | |
GCYXEGSPUDSZJY
|
6.7 | Ki | 82 | — | |
MZDKLVOWGIOKTN
|
6.7 | Ki | 80 | — | |
HPYJNDCKRXOAKV
|
6.6 | IC50 | 2 | — | |
CIBNJPAPNFXEMP
|
6.6 | IC50 | 3 | — | |
BEJCLDKQCNVTQR
|
6.6 | Ki | 16 | — |