Target Details
UniProt ACO96013
Gene SymbolPAK4
Protein NameSerine/threonine-protein kinase PAK 4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00786 (PBD) PF00069 (Pkinase)
Summary
  • Multi-target molecules 189
  • Clinical molecules 15
  • Avg pChEMBL 6.84
Top Co-occurrence Targets
Active Molecules (189)
InChIKey pChEMBL Type Targets Clinical
OWRXHGAFWZFFCW 8.8 Ki 113
QXQGBBYXXQZSKI 8.7 Ki 2
DAIDEVNNUBHVBO 8.5 Ki 2
RZXMIHOUHYSGJO 8.4 IC50 4
TUBDCTXNBUJRCI 8.4 Ki 2
NXSJMRCTGYTSTK 8.3 Kd 200
PYMVIDGHKYXJSP 8.2 IC50 2
BDWUEWMICRZPSU 8.2 Ki 2
OSVUGUHRKMMBSE 8.2 Kd 170
SFSVHJLQTWQXIO 8.2 Ki 2
HKSZLNNOFSGOKW 8.2 IC50 408
HKSZLNNOFSGOKW 8.2 Kd 213
YZRNTUZWKUDHCV 8.2 Ki 2
HKSZLNNOFSGOKW 8.1 Ki 118
KHGPYYFCIAISBU 8.1 Ki 31
RTGFZUPLFGBDKE 8.1 IC50 2
SAUMCBNMXFSRFP 8.0 Kd 2
JZTOUVBEZONDKA 8.0 Ki 80
ZKLJKKASNXVQBZ 8.0 Ki 27
DNTNKJATBLJMII 7.9 Ki 2
FBWZAFQEOKNGQL 7.8 IC50 2
MVJMMLFMPWITEJ 7.8 Ki 110
XDENYPBBMVGONB 7.8 Ki 2
FPQNRXITKTZFMF 7.8 Kd 13
KGPGFQWBCSZGEL 7.7 Kd 59 Yes
AYCPARAPKDAOEN 7.7 IC50 73
PUYIXDDMOUMMRR 7.7 Ki 27
UIARLYUEJFELEN 7.6 Kd 289 Yes
FUMCKNCUEAQHCV 7.6 Ki 103
LACOMQAWPSFXQC 7.6 Ki 27
LPILBMJJRGTKOQ 7.6 Ki 27
PBCZSGKMGDDXIJ 7.6 Kd 68 Yes
XNWKXXIGSPPPBH 7.6 Ki 31
GPOFFPKHCADYGY 7.6 Ki 2
JRLOPMVTMMPZMV 7.6 IC50 6
RTGFZUPLFGBDKE 7.5 Ki 2
DQPYZHUAILXFJI 7.5 Ki 27
FLEAYYMORDPWAJ 7.5 Ki 90
NJPWCTYVEJIQBM 7.5 Ki 72
NWMPVMMGSHXANZ 7.5 Ki 58
SLKCVFPEQGHNSI 7.5 Ki 29
ZGGIYFOLDBTZIL 7.5 Ki 27
TUBDCTXNBUJRCI 7.4 Ki 2
BGYVWFZMYBWCNY 7.4 Ki 30
WDARYLSSWBWVCU 7.4 Ki 49
SGUZXWKWTMWMCR 7.4 Ki 4
DPFLIZFLRMGXAC 7.3 Ki 2
UJBJWYNPUOLFIZ 7.3 IC50 49
LWFNQPZJAHBCBC 7.3 Ki 3
LSLPDHNUWRDOGC 7.3 Ki 25
2D structure