Target Details
| UniProt AC | O95977 |
|---|---|
| Gene Symbol | S1PR4 |
| Protein Name | Sphingosine 1-phosphate receptor 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 120
- Clinical molecules 0
- Avg pChEMBL 7.03
KEGG Pathways (3)
Active Molecules (120)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JJPKCGYTCKVOEU
|
9.0 | IC50 | 4 | — | |
MJFHVHNIHASYLI
|
8.9 | IC50 | 4 | — | |
JBPVYJJIRRUCJU
|
8.8 | IC50 | 4 | — | |
PEPDHHDQCCNILN
|
8.7 | IC50 | 4 | — | |
IJFAOCYEADEWAV
|
8.7 | IC50 | 4 | — | |
LRFKWQGGENFBFO
|
8.7 | IC50 | 5 | — | |
YRLWOUXQTIDPEK
|
8.5 | IC50 | 3 | — | |
GHQKYJKUIMNJCW
|
8.5 | IC50 | 4 | — | |
WDBMBYAFMOKUJU
|
8.4 | IC50 | 4 | — | |
RNDGTSGYNDTFOA
|
8.4 | IC50 | 4 | — | |
LXNKUNKMYYJPKD
|
8.4 | IC50 | 3 | — | |
KVYQKSXTMZHEPB
|
8.3 | IC50 | 4 | — | |
TXFZSDIRXYGOOU
|
8.3 | IC50 | 4 | — | |
WJTKHEJZIPMAKN
|
8.2 | IC50 | 4 | — | |
RMDMQWBLROBEJO
|
8.2 | IC50 | 3 | — | |
NOERNAQPKCFUKL
|
8.2 | IC50 | 4 | — | |
IILANYBHYYNGJK
|
8.1 | IC50 | 5 | — | |
IOBZROVFXAOQQI
|
8.1 | IC50 | 4 | — | |
BWCQGMDWAWERIV
|
8.0 | IC50 | 4 | — | |
GTROXDSLWCVOIS
|
7.9 | IC50 | 4 | — | |
KNLPKQCGTFMRRN
|
7.9 | IC50 | 2 | — | |
KKNUGAMJKIHACQ
|
7.8 | IC50 | 4 | — | |
KLULNXUHMWEEKT
|
7.8 | IC50 | 4 | — | |
LCRADRCUDVEFGB
|
7.8 | IC50 | 4 | — | |
LRFKWQGGENFBFO
|
7.8 | IC50 | 5 | — | |
NOMBGCXWXBTHTO
|
7.8 | IC50 | 4 | — | |
PGLFYYYVMFEVNN
|
7.8 | IC50 | 4 | — | |
NOMBGCXWXBTHTO
|
7.6 | IC50 | 4 | — | |
PGLFYYYVMFEVNN
|
7.6 | IC50 | 4 | — | |
TWNDWWAUVXKNMU
|
7.6 | IC50 | 4 | — | |
XGFCNYXSOCFJIR
|
7.6 | IC50 | 4 | — | |
YWXALJUJDPVVHS
|
7.6 | IC50 | 4 | — | |
QDDQIPUKAXBMBX
|
7.5 | Ki | 3 | — | |
DUYSYHSSBDVJSM
|
7.5 | Ki | 5 | — | |
HMJKTOOFFPXTGY
|
7.5 | IC50 | 4 | — | |
KUOMYSKEBPYIAO
|
7.5 | IC50 | 4 | — | |
DUYSYHSSBDVJSM
|
7.5 | IC50 | 6 | — | |
AKMFGWWEWTVUTP
|
7.4 | IC50 | 3 | — | |
IYOGKTIRIRHPOH
|
7.4 | IC50 | 6 | — | |
YBEAJMHMAMGKBN
|
7.3 | IC50 | 3 | — | |
PRUUCTGBHIGGOH
|
7.2 | IC50 | 4 | — | |
PGLFYYYVMFEVNN
|
7.2 | IC50 | 4 | — | |
QIPIWIXFCSCVEI
|
7.2 | IC50 | 3 | — | |
SHQNRSGKLNMHOS
|
7.2 | IC50 | 4 | — | |
XPZPTGRFTGBSAI
|
7.1 | IC50 | 4 | — | |
ZQHLJZUCUJZZRV
|
7.1 | IC50 | 4 | — | |
WECRLAZSZWCWDE
|
7.1 | IC50 | 5 | — | |
LGOMWSIGEIXWPD
|
7.0 | IC50 | 3 | — | |
QIPIWIXFCSCVEI
|
7.0 | IC50 | 3 | — | |
KARRQFDDSYYFAE
|
7.0 | IC50 | 4 | — |