Target Details
| UniProt AC | O95835 |
|---|---|
| Gene Symbol | LATS1 |
| Protein Name | Serine/threonine-protein kinase LATS1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) PF00627 (UBA) |
Summary
- Multi-target molecules 87
- Clinical molecules 7
- Avg pChEMBL 8.43
KEGG Pathways (3)
Active Molecules (87)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JHLONFVVTLRHIZ
|
8.4 | IC50 | 4 | — | |
ATBSEYKJNNUJPS
|
8.4 | IC50 | 2 | — | |
IDYBIWQRAAGTKU
|
8.4 | IC50 | 2 | — | |
NCWUWMQIMGPXQR
|
8.4 | IC50 | 2 | — | |
TWSFYAXEDIOFFN
|
8.4 | IC50 | 2 | — | |
UCTAUHCKGLOZHU
|
8.4 | IC50 | 2 | — | |
WNBNLESOAUCHBN
|
8.4 | IC50 | 2 | — | |
RQXXATOWBUCCAY
|
8.3 | IC50 | 2 | — | |
SBPQHDLJGZBWTL
|
8.2 | IC50 | 2 | — | |
ZFZNIZVNKXAOHL
|
8.1 | IC50 | 2 | — | |
CELWQJHESXUCFF
|
8.0 | IC50 | 2 | — | |
VXYPJGHKVFBNME
|
8.0 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.9 | IC50 | 408 | — | |
DKZYXHCYPUVGAF
|
7.8 | Kd | 112 | — | |
WIFZIPRZHKCGGL
|
7.6 | IC50 | 2 | — | |
IIRWNGPLJQXWFJ
|
7.6 | Kd | 21 | — | |
UIARLYUEJFELEN
|
7.5 | Kd | 289 | Yes | |
KPAQBWXRTMKVCB
|
7.5 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.4 | Kd | 213 | — | |
LOLPPWBBNUVNQZ
|
7.3 | Kd | 97 | Yes | |
IEDDDZFQZKDRBJ
|
7.2 | IC50 | 9 | — | |
KOZFSFOOLUUIGY
|
7.2 | Kd | 88 | Yes | |
MWKSRKSEWLRPBL
|
7.2 | Kd | 1075 | — | |
KGPGFQWBCSZGEL
|
7.1 | Kd | 59 | Yes | |
AYCPARAPKDAOEN
|
6.8 | Kd | 73 | — | |
FFSAICURRWPYFX
|
6.7 | IC50 | 2 | — | |
PKCDDUHJAFVJJB
|
6.7 | Kd | 13 | — | |
YFNWWNRZJGMDBR
|
6.4 | Kd | 35 | — | |
RYYNGWLOYLRZLK
|
6.4 | Kd | 45 | — | |
XZXHXSATPCNXJR
|
6.4 | Kd | 165 | Yes | |
ODPGGGTTYSGTGO
|
6.3 | Kd | 153 | — | |
FLBNLJLONKAPLR
|
6.2 | Kd | 31 | — | |
WINHZLLDWRZWRT
|
6.2 | Kd | 201 | Yes | |
CTNPALGJUAXMMC
|
6.1 | Kd | 151 | — | |
PIQCTGMSNWUMAF
|
6.0 | Kd | 137 | Yes | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |