Target Details
| UniProt AC | O95819 |
|---|---|
| Gene Symbol | MAP4K4 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 496
- Clinical molecules 34
- Avg pChEMBL 6.84
KEGG Pathways (1)
Active Molecules (496)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PSCJSWRVCKUMSL
|
6.4 | Ki | 35 | — | |
QYGMZFLXMWJYRJ
|
6.4 | Ki | 14 | — | |
RVPSPMYVDLPRIK
|
6.4 | Ki | 4 | — | |
SGHXFHRRWFLILP
|
6.4 | Ki | 29 | — | |
TVLFEDKEAOXRCZ
|
6.4 | Ki | 22 | — | |
UGHBIMSDMGHFIE
|
6.4 | Ki | 10 | — | |
URNZTLZSAVLTIZ
|
6.4 | Ki | 26 | — | |
ZAARMHXLYCHRAK
|
6.4 | Ki | 20 | — | |
ZGDYBJXDIXVTLV
|
6.4 | Ki | 54 | — | |
QHWYQHKGOYXAON
|
6.4 | IC50 | 3 | — | |
QDRFBFCKKOITJI
|
6.4 | IC50 | 2 | — | |
JQLFNUDNPNFXQP
|
6.4 | IC50 | 2 | — | |
YCYMKWLYOBLWHH
|
6.4 | IC50 | 2 | — | |
NPOADWCORNFOPY
|
6.3 | IC50 | 2 | — | |
OWWRMDBDEKIWBK
|
6.3 | IC50 | 2 | — | |
AOBLBPWPSKBHSI
|
6.3 | Ki | 55 | — | |
CACMTVGXYAZZNY
|
6.3 | Ki | 11 | — | |
CQBBMNXXVMOFCA
|
6.3 | Ki | 39 | — | |
CTJAMSGCMYAVCZ
|
6.3 | Ki | 14 | — | |
FAIHBCXQSBIRIL
|
6.3 | Ki | 22 | — | |
GHPFSYCYZJKVDZ
|
6.3 | Ki | 18 | Yes | |
GSXRCPJTNIGKSZ
|
6.3 | Ki | 43 | — | |
HDAJDNHIBCDLQF
|
6.3 | IC50 | 14 | — | |
IJRBJCMLWLFMIN
|
6.3 | Ki | 17 | — | |
IPTSYCYNQJITNJ
|
6.3 | Ki | 12 | — | |
KIUHBHFVVQQALF
|
6.3 | Ki | 9 | — | |
LRINYHMQZRENCY
|
6.3 | Ki | 29 | — | |
MQRDVGBWWVWMEN
|
6.3 | Ki | 47 | — | |
NERQMDXDVAZVNX
|
6.3 | Ki | 13 | — | |
NLDZIKOJZCTRAZ
|
6.3 | Ki | 5 | — | |
NSDIHUXUFJHXRA
|
6.3 | Ki | 11 | — | |
PEXKNSGOEOREKM
|
6.3 | Ki | 13 | — | |
SBFPHSVZEXSHTL
|
6.3 | Ki | 62 | — | |
SQXSMLLCDWJNAC
|
6.3 | Ki | 20 | — | |
UEJXQVWENDKSJQ
|
6.3 | Ki | 2 | — | |
UIRCQOKSJDLYBB
|
6.3 | Ki | 50 | — | |
XFHCSNRQFQRLHZ
|
6.3 | Ki | 12 | Yes | |
XSDJOIOVIMPMHD
|
6.3 | Ki | 44 | — | |
YDOPLCNFRXOHCC
|
6.3 | Ki | 28 | — | |
ZGZVRPRSFXRGCF
|
6.3 | Ki | 76 | — | |
VICAQGVISLDXME
|
6.3 | IC50 | 2 | — | |
FCHBYZITXHHPQO
|
6.3 | IC50 | 2 | — | |
HAMDXXRICGFPSH
|
6.2 | IC50 | 2 | — | |
BBBSTZKWEGVBNW
|
6.2 | IC50 | 2 | — | |
WCWUXEGQKLTGDX
|
6.2 | Kd | 22 | Yes | |
YRCHYHRCBXNYNU
|
6.2 | Kd | 13 | — | |
PGFXFAOPCBAZDE
|
6.2 | IC50 | 2 | — | |
GQLWKGVBOIYMTN
|
6.2 | Ki | 35 | — | |
HDRLAVNNWSHSOA
|
6.2 | Ki | 19 | — | |
HHHWHXLLZCRLAO
|
6.2 | Ki | 5 | — |