Target Details
| UniProt AC | O95819 |
|---|---|
| Gene Symbol | MAP4K4 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 496
- Clinical molecules 34
- Avg pChEMBL 6.84
KEGG Pathways (1)
Active Molecules (496)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VKQYTMVZQKCCID
|
6.6 | IC50 | 2 | — | |
IVRXNBXKWIJUQB
|
6.6 | IC50 | 10 | — | |
RVSSNRBUPQUIEG
|
6.6 | IC50 | 5 | — | |
WGDZJXGKHCWRMM
|
6.6 | IC50 | 2 | — | |
DYNHJHQFHQTFTP
|
6.5 | Kd | 38 | — | |
OYONTEXKYJZFHA
|
6.5 | Kd | 69 | Yes | |
OWAWLQLFAIHPQT
|
6.5 | IC50 | 2 | — | |
RBCWFGWXMPYQSB
|
6.5 | IC50 | 2 | — | |
HWXVIOGONBBTBY
|
6.5 | Kd | 27 | — | |
KOONCLIJVVMZCL
|
6.5 | IC50 | 2 | — | |
KXYYTXVXVOWNIG
|
6.5 | IC50 | 2 | — | |
PHXJVRSECIGDHY
|
6.5 | Kd | 59 | — | |
BJJHHKOPTKQUFQ
|
6.5 | Ki | 3 | — | |
CUIHSIWYWATEQL
|
6.5 | Ki | 61 | Yes | |
HEUSUIRCBWROMH
|
6.5 | Ki | 64 | — | |
JMQCXZBXWOIDIO
|
6.5 | Ki | 9 | — | |
KRIUNPBAQZGFQA
|
6.5 | Ki | 76 | — | |
MLGGUGPIWDHBAI
|
6.5 | Ki | 33 | — | |
MMFBBQQGBVPLQQ
|
6.5 | Ki | 13 | — | |
NXNQLECPAXXYTR
|
6.5 | Ki | 29 | — | |
ODNOTLMFNVWFTJ
|
6.5 | Ki | 11 | — | |
PAIFYAZSILXLBO
|
6.5 | Ki | 26 | — | |
QXRJBJVCBQSLTA
|
6.5 | Ki | 29 | — | |
RGOPHVZLEMGMBZ
|
6.5 | Ki | 20 | — | |
UVZVWLFSZNPMBS
|
6.5 | Ki | 17 | — | |
WYLVFMBGPRCDQF
|
6.5 | Ki | 14 | — | |
XIOOJUQFJYPVLA
|
6.5 | Ki | 17 | — | |
XJSFDMGICAWQFS
|
6.5 | Ki | 60 | — | |
XNEPVLVYFUGJLF
|
6.5 | Ki | 27 | — | |
XZWVOUQIYLZUCJ
|
6.5 | Ki | 23 | — | |
ZKHDDJKHTPLPOQ
|
6.5 | Ki | 62 | — | |
IJMQBOIQHQRHNW
|
6.5 | IC50 | 2 | — | |
NLNNYHCSSJWXLH
|
6.5 | IC50 | 2 | — | |
JWNPDZNEKVCWMY
|
6.5 | Kd | 57 | Yes | |
WVUNYSQLFKLYNI
|
6.5 | Kd | 46 | Yes | |
VHADCIRDAFWKDN
|
6.5 | IC50 | 2 | — | |
RITAVMQDGBJQJZ
|
6.5 | Kd | 43 | — | |
JKAPZPMQKNTGJW
|
6.5 | IC50 | 2 | — | |
XBAIEEJJCJHBDL
|
6.5 | Ki | 17 | — | |
MZDKLVOWGIOKTN
|
6.4 | Kd | 80 | — | |
PCPUDOGTYFUPFV
|
6.4 | IC50 | 2 | — | |
AKOITYPGORWENQ
|
6.4 | Ki | 2 | — | |
CDMGBJANTYXAIV
|
6.4 | Ki | 34 | Yes | |
GWMATETWMAQOFL
|
6.4 | Ki | 36 | — | |
JCFJQIHDZHHMQT
|
6.4 | Ki | 42 | — | |
KYACBMRLQMEIAI
|
6.4 | Ki | 30 | — | |
MFMXAWQGPQXDRJ
|
6.4 | Ki | 27 | — | |
OWFXKTOLFUQPDJ
|
6.4 | Ki | 36 | — | |
OWRXHGAFWZFFCW
|
6.4 | Ki | 113 | — | |
PQOAVBVTXNJMCM
|
6.4 | Ki | 8 | — |