Target Details
| UniProt AC | O95819 |
|---|---|
| Gene Symbol | MAP4K4 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 496
- Clinical molecules 34
- Avg pChEMBL 6.84
KEGG Pathways (1)
Active Molecules (496)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KTWBYGUSEYSRND
|
6.9 | Ki | 28 | — | |
MULNSLQVKKUPJN
|
6.9 | Ki | 41 | — | |
ONSQVIFJAFIKFZ
|
6.9 | Ki | 6 | — | |
QONPPIZSNSSCSK
|
6.9 | Ki | 45 | Yes | |
XBNSDTLFWKORGH
|
6.9 | Ki | 10 | — | |
XLSYZSRXVVCHLS
|
6.9 | Kd | 48 | — | |
YXTUXFBKHGBPPN
|
6.9 | IC50 | 2 | — | |
CPSFZCLACXEMLI
|
6.9 | IC50 | 2 | — | |
JCOMWFYBHHOUGK
|
6.9 | IC50 | 2 | — | |
KHPCIHZXOGHCLY
|
6.9 | IC50 | 3 | — | |
YLDDOLAWPICWDH
|
6.9 | IC50 | 2 | — | |
BPNUQXPIQBZCMR
|
6.8 | Kd | 83 | Yes | |
GUBJNPWVIUFSTR
|
6.8 | Kd | 103 | — | |
PEOZMOGNFLONKU
|
6.8 | IC50 | 2 | — | |
TZMCWEXCNHTWOP
|
6.8 | IC50 | 2 | — | |
WINHZLLDWRZWRT
|
6.8 | Kd | 201 | Yes | |
XZXHXSATPCNXJR
|
6.8 | Kd | 165 | Yes | |
AQZIXHSRFOGYHF
|
6.8 | Ki | 9 | — | |
DJLORVJVWIBDME
|
6.8 | Ki | 24 | — | |
DWXUTKBSWVUPBE
|
6.8 | Ki | 8 | — | |
HSMUWLLZAZCLHF
|
6.8 | Ki | 25 | — | |
HXHAJRMTJXHJJZ
|
6.8 | Ki | 52 | Yes | |
JTRNNNVASYCTLO
|
6.8 | Ki | 14 | — | |
MQAKXLBEDXFDMV
|
6.8 | Ki | 5 | — | |
NHFDRBXTEDBWCZ
|
6.8 | Ki | 41 | — | |
OAVGBZOFDPFGPJ
|
6.8 | Ki | 42 | Yes | |
OEEGUWWPGAZRIJ
|
6.8 | Ki | 21 | — | |
OWFLADWRSCINST
|
6.8 | Ki | 30 | — | |
PIQCTGMSNWUMAF
|
6.8 | Kd | 137 | Yes | |
PQNWNVWJXPSZFR
|
6.8 | Ki | 21 | — | |
QTQUAHGXBLFSCH
|
6.8 | Ki | 10 | — | |
RGNHKJWHFIPHIM
|
6.8 | Ki | 66 | — | |
RITAVMQDGBJQJZ
|
6.8 | Ki | 33 | — | |
RWKDVIAVTRRJIR
|
6.8 | Ki | 23 | — | |
SKKRZILJUKYLJS
|
6.8 | Ki | 25 | — | |
SRROIPFGGDHJCJ
|
6.8 | Ki | 7 | — | |
UHTHHESEBZOYNR
|
6.8 | Ki | 66 | Yes | |
UYGYYOIUVFMGKQ
|
6.8 | Ki | 30 | — | |
XVUSMHCLFMFBQR
|
6.8 | IC50 | 3 | — | |
XXSPHNFKLDJDAK
|
6.8 | Ki | 26 | — | |
ZLVOTRRGLSDLPF
|
6.8 | Ki | 36 | — | |
AMTPPKYFTXUVJY
|
6.8 | IC50 | 2 | — | |
VLPQFOXQPCFHRL
|
6.8 | IC50 | 2 | — | |
OWRPRNROGDZURV
|
6.8 | IC50 | 2 | — | |
AVEXLWXITHDXGJ
|
6.8 | IC50 | 2 | — | |
MWTNEWVBVSRDNA
|
6.8 | IC50 | 2 | — | |
GOYOZLWEHBWSHT
|
6.7 | IC50 | 2 | — | |
CXQHYVUVSFXTMY
|
6.7 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.7 | Kd | 149 | — | |
WCCMSFLKQHUQAF
|
6.7 | IC50 | 2 | — |