Target Details
| UniProt AC | O95819 |
|---|---|
| Gene Symbol | MAP4K4 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 496
- Clinical molecules 34
- Avg pChEMBL 6.84
KEGG Pathways (1)
Active Molecules (496)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MZIOLOXGGOLJMJ
|
7.1 | Ki | 12 | — | |
TVUWQDLBEOZVOU
|
7.1 | Ki | 41 | — | |
VEXYJVKMGKPGRV
|
7.1 | Ki | 6 | — | |
VOAZYSSSBBQYMU
|
7.1 | Ki | 4 | — | |
VUHZDNOPEVGHEO
|
7.1 | Ki | 29 | — | |
VYACUCWGDYRIAG
|
7.1 | Ki | 7 | — | |
YJVZYDNNGQCFEQ
|
7.1 | IC50 | 2 | — | |
DKZYXHCYPUVGAF
|
7.1 | Kd | 112 | — | |
VEMZDHGGFCZOTO
|
7.1 | IC50 | 2 | — | |
MVCOAUNKQVWQHZ
|
7.0 | Kd | 54 | Yes | |
SENWNDLDAHBDSA
|
7.0 | IC50 | 2 | — | |
UADCTKCTCBTSLU
|
7.0 | IC50 | 2 | — | |
GYOQXOATKFOYNW
|
7.0 | IC50 | 2 | — | |
RBPNVVLVIGSUDX
|
7.0 | IC50 | 2 | — | |
ROBNMKKERIMYQP
|
7.0 | IC50 | 2 | — | |
ACSYKUPGCXYRRO
|
7.0 | Ki | 26 | — | |
ADLPKFFMGIJZIM
|
7.0 | Ki | 44 | — | |
CJNRNQUPGPBLID
|
7.0 | IC50 | 2 | — | |
GVOOEMLKTIRYCO
|
7.0 | Ki | 7 | — | |
IZAVTOABECKIDH
|
7.0 | Ki | 20 | — | |
JTRXEPCDEVNYPE
|
7.0 | Ki | 5 | — | |
JWQOJVOKBAAAAR
|
7.0 | Ki | 29 | — | |
MCCCQFAOMZMZKE
|
7.0 | Ki | 52 | — | |
QPORZABOFXPRHM
|
7.0 | Ki | 18 | — | |
QRCXMLQLNQMAFC
|
7.0 | Ki | 10 | — | |
QXKKPVVOOWBLND
|
7.0 | Ki | 8 | — | |
RYYNGWLOYLRZLK
|
7.0 | Ki | 104 | — | |
SRUYMJRFVGLQDV
|
7.0 | Ki | 37 | — | |
VUWOSKCPLJROAK
|
7.0 | Ki | 6 | — | |
XHORJSJFHVABEA
|
7.0 | Ki | 49 | — | |
RUHNYDZQGMWRMX
|
7.0 | IC50 | 2 | — | |
VHBIVOIWMNXHQR
|
7.0 | IC50 | 2 | — | |
PAZJYAQBBSYLRQ
|
7.0 | IC50 | 2 | — | |
FTBRALICGUIRHO
|
7.0 | IC50 | 2 | — | |
KNAKHJWNZMAMAO
|
7.0 | IC50 | 2 | — | |
LOLPPWBBNUVNQZ
|
7.0 | Kd | 97 | Yes | |
OYWNKAAPXTYEBN
|
7.0 | IC50 | 6 | — | |
KSOOWLORAVQWKJ
|
7.0 | IC50 | 2 | — | |
OOSMLYPLUCBANZ
|
7.0 | IC50 | 2 | — | |
UBPYMWXTLXKKBW
|
7.0 | IC50 | 2 | — | |
VKBFHTIUXUCYRQ
|
7.0 | Ki | 66 | — | |
LQYGLUICAZYCHN
|
6.9 | IC50 | 2 | — | |
MGTQMPVMKHKJAF
|
6.9 | IC50 | 2 | — | |
YFZOGSFWULXJTA
|
6.9 | IC50 | 2 | — | |
MPUBMJCSEANNKB
|
6.9 | IC50 | 2 | — | |
SQKBBDOFPPNVCL
|
6.9 | IC50 | 4 | — | |
ULMJOBGKUKPBKO
|
6.9 | IC50 | 2 | — | |
BIFCETOSTFEUQU
|
6.9 | IC50 | 2 | — | |
CLEGDJQQHUTCOW
|
6.9 | Ki | 43 | — | |
GCBJDOWIQHMCMR
|
6.9 | Ki | 84 | — |