Target Details
| UniProt AC | O95819 |
|---|---|
| Gene Symbol | MAP4K4 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 496
- Clinical molecules 34
- Avg pChEMBL 6.84
KEGG Pathways (1)
Active Molecules (496)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZKLJKKASNXVQBZ
|
7.4 | Ki | 27 | — | |
ZQUSFAUAYSEREK
|
7.4 | Ki | 7 | — | |
CLODUYRNZMIONW
|
7.4 | IC50 | 3 | — | |
QACLFFVLWCKNEA
|
7.4 | IC50 | 2 | — | |
MSWOWUREQODTRO
|
7.4 | IC50 | 11 | — | |
NETVGXQSFUMKOX
|
7.4 | IC50 | 2 | — | |
WVXNSAVVKYZVOE
|
7.3 | IC50 | 92 | — | |
GOUXACDXZWAKJI
|
7.3 | IC50 | 2 | — | |
CNQGNADBGYCKKV
|
7.3 | Ki | 25 | — | |
DFMCXVONDDGQIY
|
7.3 | Ki | 66 | — | |
HOYRWTWZUFFACV
|
7.3 | Ki | 28 | — | |
IORLJCFZTVIEHA
|
7.3 | IC50 | 2 | — | |
JZTOUVBEZONDKA
|
7.3 | Ki | 80 | — | |
NFMGZVPRGVERNN
|
7.3 | Ki | 44 | — | |
NZVDDFRUBIEKLV
|
7.3 | Ki | 20 | — | |
QNUKRWAIZMBVCU
|
7.3 | Ki | 46 | — | |
UUWNXFJBBYAMDT
|
7.3 | Ki | 46 | — | |
WPHKIQPVPYJNAX
|
7.3 | Ki | 81 | — | |
XBTZKVHEBBNOCK
|
7.3 | IC50 | 2 | — | |
XKZINYYXWJEYEL
|
7.3 | Ki | 37 | — | |
XKZQZMSAWVDRSP
|
7.3 | Ki | 39 | Yes | |
XSRHBCYNCKAFKS
|
7.3 | Ki | 45 | — | |
YWTBGJGMTBHQTM
|
7.3 | Ki | 65 | — | |
ZWVZORIKUNOTCS
|
7.3 | Ki | 69 | — | |
WWFSKAMRQLRLTJ
|
7.3 | IC50 | 2 | — | |
ACHHYBWZGKASQH
|
7.2 | IC50 | 2 | — | |
MGHJYWHFIWPSNB
|
7.2 | IC50 | 2 | — | |
ADMFLILDQJSEIK
|
7.2 | Ki | 72 | — | |
AZTMYWWWILJAKW
|
7.2 | Ki | 16 | Yes | |
HSXHOPFVRFPEGS
|
7.2 | IC50 | 2 | — | |
HZGYSSZTTMUCJE
|
7.2 | Ki | 8 | — | |
IAKGNUWZPSPEKU
|
7.2 | Ki | 19 | — | |
MHCPAORAYMTGCZ
|
7.2 | Ki | 37 | — | |
MVJMMLFMPWITEJ
|
7.2 | Ki | 110 | — | |
OUORNBBPANSKFS
|
7.2 | Ki | 3 | — | |
UAQJVFADAYIBGC
|
7.2 | Ki | 23 | — | |
VQPBIJGXSXEOCU
|
7.2 | Ki | 24 | — | |
YMIJUBCSOKSFRU
|
7.2 | Ki | 87 | — | |
YMSZHISTTIUBDG
|
7.2 | Ki | 7 | — | |
YUOWJICKAJQZLS
|
7.2 | Ki | 35 | — | |
CXMURJVCMJRHAM
|
7.2 | IC50 | 2 | — | |
WNEVOMUAXQPYDE
|
7.2 | IC50 | 2 | — | |
WTYJCTRCRZLZFE
|
7.2 | IC50 | 2 | — | |
AIYREGHPXFOWSK
|
7.2 | IC50 | 2 | — | |
LXGDXFKSYPYLSD
|
7.1 | IC50 | 2 | — | |
CTQIQHVVPQICIK
|
7.1 | Ki | 7 | — | |
CYLYPHIGBMPKCK
|
7.1 | Ki | 6 | — | |
DQPYZHUAILXFJI
|
7.1 | Ki | 27 | — | |
IFPPYSWJNWHOLQ
|
7.1 | Ki | 52 | Yes | |
IJNGXROUMFEKDB
|
7.1 | Ki | 39 | — |