Target Details
| UniProt AC | O95819 |
|---|---|
| Gene Symbol | MAP4K4 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 496
- Clinical molecules 34
- Avg pChEMBL 6.84
KEGG Pathways (1)
Active Molecules (496)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SDBOIBYRBWPIEL
|
7.7 | Ki | 31 | — | |
UDFDIIVNIYWXDM
|
7.7 | Ki | 74 | — | |
WDARYLSSWBWVCU
|
7.7 | Ki | 49 | — | |
XOJQJDHWKVZUAT
|
7.7 | Ki | 9 | — | |
ZYTFPHRVOZXPGZ
|
7.7 | Ki | 30 | — | |
XFEKSSMJINNJSX
|
7.7 | IC50 | 3 | — | |
VBQRUKZVDRXMBF
|
7.7 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
7.6 | Kd | 289 | Yes | |
HKSZLNNOFSGOKW
|
7.6 | Kd | 213 | — | |
MHEOXLMQZIYGDG
|
7.6 | IC50 | 2 | — | |
CXBBWVXSZINRCS
|
7.6 | Ki | 41 | — | |
HEKAIDKUDLCBRU
|
7.6 | Ki | 20 | — | |
KARJFNUGCLEZKM
|
7.6 | IC50 | 3 | — | |
KWRXWPRFIUJQBP
|
7.6 | Ki | 25 | — | |
OFPXYNMQWVCVKZ
|
7.6 | Ki | 8 | — | |
PLHUMPJXRHMFFR
|
7.6 | Ki | 28 | — | |
RFBPWKMQWSIPEO
|
7.6 | Ki | 28 | — | |
VCFDMLBPASGZTP
|
7.6 | Ki | 38 | — | |
XJJYJNMNYDNXNO
|
7.6 | Ki | 23 | — | |
FJICSOOOGVNUCL
|
7.5 | IC50 | 2 | — | |
QABFDCSQZQSQOW
|
7.5 | IC50 | 2 | — | |
YDBNEDDJBRLASN
|
7.5 | IC50 | 2 | — | |
CEOYEZFCROSXBX
|
7.5 | IC50 | 2 | — | |
KQBUVBWQFHWPMI
|
7.5 | IC50 | 2 | — | |
GDYZFFBMSBDTAA
|
7.5 | Ki | 60 | — | |
KBDRSPRFXNCQAM
|
7.5 | Ki | 8 | — | |
LXSCQGMBFODPHP
|
7.5 | IC50 | 2 | — | |
RBXYGQNZRVPDNB
|
7.5 | Ki | 34 | — | |
VLEFVPMCVJDTHZ
|
7.5 | Ki | 13 | — | |
WINHZLLDWRZWRT
|
7.5 | Ki | 66 | — | |
XOOAAYRIVATZNM
|
7.5 | Ki | 55 | — | |
XPHWIERLJBFPFV
|
7.5 | Ki | 69 | — | |
YYLKKYCXAOBSRM
|
7.5 | Kd | 191 | — | |
APXIUBHZWNOTAS
|
7.5 | IC50 | 2 | — | |
IAYGCINLNONXHY
|
7.5 | Kd | 50 | — | |
VHADCIRDAFWKDN
|
7.4 | IC50 | 2 | — | |
ISSFPHPDMLUKPK
|
7.4 | IC50 | 2 | — | |
AGYZUONRISUOIK
|
7.4 | Ki | 10 | — | |
AUDNGNGLLRZLDR
|
7.4 | Ki | 33 | — | |
GHMRUNOHAHJNNA
|
7.4 | Ki | 29 | — | |
JSDGKSMNPHJDFK
|
7.4 | Ki | 35 | — | |
KHGPYYFCIAISBU
|
7.4 | Ki | 31 | — | |
NBLFGELIWIKRAC
|
7.4 | Ki | 8 | — | |
NLUPJKQOKWBWFC
|
7.4 | Ki | 69 | — | |
OLUKILHGKRVDCT
|
7.4 | Ki | 44 | Yes | |
PNKALLUVKOKYHZ
|
7.4 | Ki | 32 | — | |
XNWKXXIGSPPPBH
|
7.4 | Ki | 31 | — | |
XUFLBSMTYMFOQH
|
7.4 | Ki | 43 | — | |
YDWMUCKJUNLURC
|
7.4 | Ki | 24 | — | |
YEHCNYAQEBQCCS
|
7.4 | Ki | 74 | — |