Target Details
| UniProt AC | O95819 |
|---|---|
| Gene Symbol | MAP4K4 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 496
- Clinical molecules 34
- Avg pChEMBL 6.84
KEGG Pathways (1)
Active Molecules (496)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SDTHQOXRWZXTJF
|
6.1 | Ki | 16 | — | |
SELXDFVNFMEQCP
|
6.1 | Ki | 5 | — | |
SFPWNTQWFFNJIH
|
6.1 | Ki | 48 | — | |
UCOWZARZLHNDKP
|
6.1 | Ki | 8 | — | |
UTQPKPHUIMHAAN
|
6.1 | Ki | 22 | — | |
VNGYQBMDQMDALH
|
6.1 | Ki | 25 | — | |
VSPFURGQAYMVAN
|
6.1 | Ki | 17 | — | |
VSVWQTDDGQSGHP
|
6.1 | Ki | 51 | — | |
WKEYMNLZBZKLOG
|
6.1 | Ki | 14 | — | |
WNTAZUFBXXQBAO
|
6.1 | Ki | 2 | — | |
XCHWBXBDZRJVDP
|
6.1 | Ki | 51 | — | |
YGUMGYOBTNGZKS
|
6.1 | Ki | 12 | — | |
YKJSWMAVAKRUAN
|
6.1 | Ki | 19 | — | |
GGQCIOOSELPMBB
|
6.1 | IC50 | 3 | — | |
GZMVECPBSUHMMJ
|
6.1 | IC50 | 3 | — | |
RTJQABCNNLMCJF
|
6.1 | IC50 | 3 | — | |
PBCZSGKMGDDXIJ
|
6.1 | Kd | 68 | Yes | |
NGDXEOHYWJHBTJ
|
6.1 | IC50 | 5 | — | |
VAARYSWULJUGST
|
6.1 | Kd | 119 | Yes | |
NAIUXUTZYFPOIK
|
6.0 | IC50 | 2 | — | |
UJBJWYNPUOLFIZ
|
6.0 | IC50 | 49 | — | |
JTVBXQAYBIJXRP
|
6.0 | Kd | 20 | — | |
QQWUGDVOUVUTOY
|
6.0 | Kd | 231 | Yes | |
CYLGCMABIBXHIQ
|
6.0 | Ki | 16 | — | |
CZIGMBNEFWBEMD
|
6.0 | Ki | 16 | — | |
DKSNLQYRZJKYOC
|
6.0 | Ki | 51 | — | |
GEGCXGMFUYJULA
|
6.0 | Ki | 30 | Yes | |
GKODJBVKKLQMEY
|
6.0 | Ki | 10 | — | |
HKZKELVPGXJIMW
|
6.0 | Ki | 41 | — | |
IGGNAIYXGIUMQZ
|
6.0 | Ki | 5 | — | |
JGKVEXCUPFIDIE
|
6.0 | Ki | 5 | — | |
JOIUJUJSHIHBDT
|
6.0 | Ki | 18 | — | |
KAKGFGCTONHQJW
|
6.0 | Ki | 25 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KJVWCDAPVMWKLJ
|
6.0 | Ki | 20 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MMMPFWNSQKXKDX
|
6.0 | Ki | 14 | — | |
QHKYPYXTTXKZST
|
6.0 | Ki | 28 | — | |
TUJUZVJICDSNLY
|
6.0 | Ki | 19 | — | |
UOOFSEUSROQBBP
|
6.0 | Ki | 8 | — | |
UTFXYGYVDDLJER
|
6.0 | Ki | 36 | — | |
WQFGNANQTYLQBP
|
6.0 | Ki | 16 | — | |
XFCOCCMXXFTEEC
|
6.0 | Ki | 6 | — | |
XGALLCVXEZPNRQ
|
6.0 | Ki | 39 | Yes | |
ZFGXZJKLOFCECI
|
6.0 | Ki | 5 | — | |
ZQVQTUFEKLITNT
|
6.0 | Ki | 10 | — |