Target Details
| UniProt AC | O95747 |
|---|---|
| Gene Symbol | OXSR1 |
| Protein Name | Serine/threonine-protein kinase OSR1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12202 (OSR1_C) PF00069 (Pkinase) |
Summary
- Multi-target molecules 6
- Clinical molecules 2
- Avg pChEMBL 6.33
KEGG Pathways (1)
Active Molecules (6)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QQWUGDVOUVUTOY
|
7.3 | Kd | 231 | Yes | |
HKSZLNNOFSGOKW
|
6.4 | Kd | 408 | — | |
WINHZLLDWRZWRT
|
6.3 | Kd | 201 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |