Target Details
| UniProt AC | O95696 |
|---|---|
| Gene Symbol | BRD1 |
| Protein Name | Bromodomain-containing protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00439 (Bromodomain) PF10513 (EPL1) PF13831 (PHD_2) PF00855 (PWWP) PF13832 (zf-HC5HC2H_2) |
Summary
- Multi-target molecules 44
- Clinical molecules 0
- Avg pChEMBL 6.79
Active Molecules (44)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HYQBRUSSCIAOOD
|
7.9 | Kd | 6 | — | |
YDDKRKCQSIKAJD
|
7.3 | IC50 | 3 | — | |
ZIQDIXVWQPULTM
|
7.2 | IC50 | 2 | — | |
LLHGUSJJGJYSJO
|
7.2 | IC50 | 2 | — | |
OFWWWKWUCDUISA
|
7.2 | IC50 | 3 | — | |
LGZFUXSDGGGPHG
|
7.2 | IC50 | 2 | — | |
LQDXWIYREJVTTB
|
7.1 | IC50 | 4 | — | |
XWUSNMULJMQCCC
|
7.1 | IC50 | 3 | — | |
OFZUZFZNFMUNAS
|
7.0 | IC50 | 3 | — | |
AHCZNZBUHSRPCU
|
7.0 | IC50 | 2 | — | |
NZCCNFWSBAAKSI
|
7.0 | IC50 | 3 | — | |
XULQOMADHZABKB
|
7.0 | IC50 | 3 | — | |
MYIGQQDEMVIHBG
|
7.0 | IC50 | 2 | — | |
UEMQPCYDWCSVCU
|
7.0 | IC50 | 5 | — | |
VZAFGXCWAWRULT
|
7.0 | Ki | 7 | — | |
NMRMIPFJPBQHHY
|
6.9 | IC50 | 2 | — | |
ZJQVEQKLMMZDON
|
6.9 | IC50 | 2 | — | |
XHAYAQCABOVSNX
|
6.9 | Kd | 9 | — | |
QFOYNDFIBXQVIO
|
6.9 | IC50 | 3 | — | |
BXGJNRVCUDKEGW
|
6.8 | IC50 | 2 | — | |
JJGHZALDUUMGCU
|
6.8 | IC50 | 3 | — | |
WUCKMZXHDIJUHE
|
6.8 | IC50 | 2 | — | |
WMKFJDQPAVKQAQ
|
6.8 | IC50 | 3 | — | |
UCCATIJMEOLTEL
|
6.8 | IC50 | 2 | — | |
YPOOJPDFTKZDEW
|
6.7 | IC50 | 3 | — | |
AMEZIZUFNQNCRU
|
6.7 | IC50 | 2 | — | |
VXXXPCKZPJGNGK
|
6.7 | IC50 | 4 | — | |
BMVCSXFOQPYKKC
|
6.7 | IC50 | 5 | — | |
GGJRFYLWAXMCNR
|
6.7 | IC50 | 2 | — | |
GPMNHYJTFYQIDD
|
6.6 | IC50 | 2 | — | |
KZNDNGJCFUTVMP
|
6.6 | IC50 | 2 | — | |
MQQWUSICUOGGBD
|
6.6 | IC50 | 2 | — | |
WNTOXMAGPDYDCR
|
6.6 | IC50 | 3 | — | |
COVNONZQYCHIJS
|
6.6 | IC50 | 2 | — | |
LIGPIGAGCDCBGQ
|
6.6 | IC50 | 2 | — | |
UQJAUEXASXFSKA
|
6.4 | IC50 | 2 | — | |
FFVNHKQONMKRRU
|
6.4 | IC50 | 2 | — | |
BTTCKSLDCMBUAH
|
6.4 | Ki | 7 | — | |
NQBBGPWFKFVWGM
|
6.4 | IC50 | 3 | — | |
HHQVWOAKOPBQDP
|
6.3 | IC50 | 2 | — | |
YUNQZQREIHWDQT
|
6.3 | Kd | 2 | — | |
BINBUXZIKUNKAE
|
6.3 | IC50 | 2 | — | |
NCCGOWLXEQZIMX
|
6.3 | IC50 | 2 | — | |
QCIJLRJBZDBVDB
|
6.1 | Kd | 5 | — |