Target Details
| UniProt AC | O95382 |
|---|---|
| Gene Symbol | MAP3K6 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF19039 (ASK_PH) PF20309 (DRHyd-ASK) PF20302 (HisK-N-like) PF13281 (MAP3K_TRAF_bd) PF00069 (Pkinase) |
Summary
- Multi-target molecules 11
- Clinical molecules 2
- Avg pChEMBL 7.04
KEGG Pathways (1)
Active Molecules (11)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GXPOETDGLYYIAQ
|
8.2 | IC50 | 2 | — | |
MUAQRESRLYYNEV
|
8.1 | IC50 | 2 | — | |
LUQKIXFXOFQGGI
|
7.8 | IC50 | 2 | — | |
ZLOBOPFIUGIVMK
|
7.8 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
6.8 | Kd | 289 | Yes | |
FKDNUEBNRIFBDZ
|
6.7 | IC50 | 3 | — | |
ANCZNPGQXFLAIW
|
6.6 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
6.6 | IC50 | 408 | — | |
KOZFSFOOLUUIGY
|
6.5 | Kd | 88 | Yes | |
SMJAMOAYGIVKRI
|
6.3 | IC50 | 4 | — | |
UBSRPCYTKJDJKN
|
6.1 | IC50 | 2 | — |