Target Details
| UniProt AC | O95271 |
|---|---|
| Gene Symbol | TNKS |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 711
- Clinical molecules 0
- Avg pChEMBL 7.76
Active Molecules (711)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WFJABTXVQUHYJP
|
7.7 | IC50 | 3 | — | |
WWOMDTSWLDXWQW
|
7.7 | IC50 | 2 | — | |
XHBUHAYJGXCPDR
|
7.7 | IC50 | 2 | — | |
GERFIVKNGYXTHK
|
7.7 | IC50 | 2 | — | |
MCCQXQRJNJXHRG
|
7.7 | IC50 | 3 | — | |
TYQINFQXCFVKCF
|
7.7 | IC50 | 2 | — | |
GXKPLMIZTNQPMI
|
7.6 | IC50 | 2 | — | |
IGKALBMMBUOLAY
|
7.6 | IC50 | 2 | — | |
XAQYIMOAZYNCLU
|
7.6 | IC50 | 2 | — | |
YXOMGSWERMJJSE
|
7.6 | IC50 | 2 | — | |
IAIXKHJSBQJCKK
|
7.6 | IC50 | 2 | — | |
NEUUVLLFIFUTLB
|
7.6 | IC50 | 2 | — | |
QOUNQNYSBYTMLY
|
7.6 | IC50 | 2 | — | |
VLKQIEMXMFAOES
|
7.6 | IC50 | 2 | — | |
WPCRHWQMOWNQPY
|
7.6 | IC50 | 2 | — | |
WPVANBBTWUUEFL
|
7.6 | IC50 | 2 | — | |
BVKOWESRQTZUCM
|
7.6 | IC50 | 2 | — | |
DTOVAHAAYGWZJC
|
7.6 | IC50 | 2 | — | |
MPGRGIIZXCNTKV
|
7.6 | IC50 | 2 | — | |
PVUNOEJZLPVTPG
|
7.6 | IC50 | 2 | — | |
HWSBIYJZGFCBGQ
|
7.6 | IC50 | 2 | — | |
VFXBLJYICQUSGU
|
7.6 | IC50 | 2 | — | |
YBDVEUNJLWDATQ
|
7.6 | IC50 | 2 | — | |
ZEQVKZNUMQSOLV
|
7.6 | IC50 | 2 | — | |
DBNHRWOXIIAGGS
|
7.6 | IC50 | 2 | — | |
DDIZJESACWEABB
|
7.6 | IC50 | 2 | — | |
HIXCMHOBVDTAIE
|
7.6 | IC50 | 2 | — | |
RDAGLFLFHKNHGG
|
7.6 | IC50 | 2 | — | |
SJXSPWSYROZIMI
|
7.6 | IC50 | 2 | — | |
SOKUIQBGUJNMGO
|
7.6 | IC50 | 2 | — | |
HWGQMRYQVZSGDQ
|
7.6 | Kd | 7 | — | |
CDZVLUPXXHOPPI
|
7.5 | IC50 | 2 | — | |
GNNYYUFPAQKZRD
|
7.5 | IC50 | 2 | — | |
ULCIOMUEHZHNQU
|
7.5 | IC50 | 2 | — | |
XTWGYPAWWDNGTC
|
7.5 | IC50 | 3 | — | |
ZAVBKFISCRSHAT
|
7.5 | IC50 | 2 | — | |
GWIUFTNKTNCPNA
|
7.5 | IC50 | 2 | — | |
IEJZGHYRQZYUPZ
|
7.5 | IC50 | 2 | — | |
MFDYBTCPKCGNLY
|
7.5 | IC50 | 2 | — | |
MYNRZMIPPXBMLY
|
7.5 | IC50 | 2 | — | |
RJIONECKTUPQGG
|
7.5 | IC50 | 2 | — | |
SBYKJNMYJXVHLX
|
7.5 | IC50 | 2 | — | |
XSXNSAZKDIVZTL
|
7.5 | IC50 | 2 | — | |
JJHZDQRUCBOSIK
|
7.5 | IC50 | 3 | — | |
LJLQEWDFIMKBSL
|
7.5 | IC50 | 2 | — | |
MXRLSJYSHPXDBN
|
7.5 | IC50 | 2 | — | |
WTVLTJMRTHFMJP
|
7.5 | IC50 | 2 | — | |
XGTNOTWEBRRAKO
|
7.5 | IC50 | 2 | — | |
BCVWBJPQPDBXMM
|
7.5 | IC50 | 3 | — | |
DBBRJAYFAWANIO
|
7.5 | IC50 | 2 | — |