Target Details
| UniProt AC | O95271 |
|---|---|
| Gene Symbol | TNKS |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 711
- Clinical molecules 0
- Avg pChEMBL 7.76
Active Molecules (711)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FXPQKIUFVMHDMQ
|
7.8 | IC50 | 2 | — | |
HRUWZYLXSAQFEL
|
7.8 | IC50 | 2 | — | |
KCPHCJUACXXHDI
|
7.8 | IC50 | 2 | — | |
PQGLPXUXVBAMGX
|
7.8 | IC50 | 2 | — | |
BTVYOOANNCDQKM
|
7.8 | IC50 | 2 | — | |
FVSMOECHMBICED
|
7.8 | IC50 | 3 | — | |
KVVODYVRKLLEIQ
|
7.8 | IC50 | 2 | — | |
PSUPASCETWCMMJ
|
7.8 | IC50 | 2 | — | |
REUQDXNRIHMJKE
|
7.8 | IC50 | 2 | — | |
SDDYULNTURKZSO
|
7.8 | IC50 | 2 | — | |
WZAAURATTBNWBC
|
7.8 | IC50 | 2 | — | |
DYGBNAYFDZEYBA
|
7.8 | IC50 | 3 | — | |
SUKHPNUTRMBUST
|
7.8 | IC50 | 4 | — | |
ADXVPUDCPCBXPZ
|
7.8 | IC50 | 2 | — | |
GVSKTDUUGXDISO
|
7.8 | IC50 | 2 | — | |
HDPKFKWBVMIZEB
|
7.8 | IC50 | 2 | — | |
HXWKRLPCYVNDNE
|
7.8 | IC50 | 2 | — | |
KGBRRRXNQADTEZ
|
7.8 | IC50 | 2 | — | |
PAMUWGVDNNJVJY
|
7.8 | IC50 | 2 | — | |
WMCHACNVSFKECE
|
7.8 | IC50 | 2 | — | |
AMYVNCAWBFVJCR
|
7.8 | IC50 | 2 | — | |
WRWWRQVRBZBWSL
|
7.8 | IC50 | 3 | — | |
KBKQSDRVJSIUST
|
7.8 | IC50 | 2 | — | |
KMMKOGNMTHXBIM
|
7.8 | IC50 | 2 | — | |
KMOJQLGIBUUKKE
|
7.8 | IC50 | 2 | — | |
LANJYZWTSUUASB
|
7.8 | IC50 | 3 | — | |
SVDUOSYBBYZAAB
|
7.8 | IC50 | 2 | — | |
UHPJRQMZYNOZHL
|
7.8 | IC50 | 2 | — | |
ZPMJHPPAFDZXFG
|
7.8 | IC50 | 2 | — | |
FSNRYQUQAYKAPH
|
7.8 | IC50 | 4 | — | |
HMUTYRXLOPTZOV
|
7.8 | IC50 | 2 | — | |
LTQNPKURAUAWPU
|
7.8 | IC50 | 2 | — | |
WLVFPFBPOHXOMK
|
7.8 | IC50 | 2 | — | |
CLMCMCIANXSSCI
|
7.7 | IC50 | 2 | — | |
FOMOQTCFXCTELV
|
7.7 | IC50 | 2 | — | |
ULCGWFIERYSNSV
|
7.7 | IC50 | 2 | — | |
WDZBHMSPANOWRC
|
7.7 | IC50 | 2 | — | |
ZNAKJYRBQMWNHT
|
7.7 | IC50 | 2 | — | |
BVBKPRYPLQAWKE
|
7.7 | IC50 | 3 | — | |
ZKOSRIBDKQNGTM
|
7.7 | IC50 | 2 | — | |
FOFNXWJHZNRHCH
|
7.7 | IC50 | 2 | — | |
RBDQSAKXGCRFGL
|
7.7 | IC50 | 2 | — | |
DKYAMBSWXNVNIR
|
7.7 | IC50 | 2 | — | |
DUCZLEBAUSAZOC
|
7.7 | IC50 | 2 | — | |
QWQWNLQBJNFADI
|
7.7 | IC50 | 2 | — | |
MFVKIQGUHZYYOF
|
7.7 | IC50 | 2 | — | |
PRPXVBJXNFAFSR
|
7.7 | IC50 | 2 | — | |
OQNRYQMRIGYPGK
|
7.7 | IC50 | 2 | — | |
UTGVEYXWHNPJKF
|
7.7 | IC50 | 3 | — | |
WAYVCDVUNSIWJI
|
7.7 | IC50 | 2 | — |