Target Details
| UniProt AC | O95271 |
|---|---|
| Gene Symbol | TNKS |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 711
- Clinical molecules 0
- Avg pChEMBL 7.76
Active Molecules (711)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZDDPBFWHZOJFHF
|
8.1 | IC50 | 6 | — | |
HILQRGHXDPSDBM
|
8.0 | IC50 | 2 | — | |
JMJMHZKQKKROFG
|
8.0 | IC50 | 2 | — | |
YXSXXZZWNFHIGM
|
8.0 | IC50 | 2 | — | |
FICOSMQGCGGNKM
|
8.0 | IC50 | 2 | — | |
NVYDBKBQXGPVQD
|
8.0 | IC50 | 2 | — | |
XIFIENIKEZUQQD
|
8.0 | IC50 | 2 | — | |
VXRWQCMYTRYKQD
|
8.0 | IC50 | 2 | — | |
XPFCXDCYIAOOBE
|
8.0 | IC50 | 2 | — | |
FHBYLOWAINBPRJ
|
8.0 | IC50 | 4 | — | |
IKPHQSQQUCQZBC
|
8.0 | IC50 | 2 | — | |
ILBZVTXOJSVUIM
|
8.0 | IC50 | 2 | — | |
QIVMBVYEEIHHKY
|
8.0 | IC50 | 2 | — | |
UXGMDGPWMVIMFP
|
8.0 | IC50 | 2 | — | |
KXVJOZBQCTUYNT
|
8.0 | IC50 | 2 | — | |
FDLYAMZZIXQODN
|
8.0 | IC50 | 11 | — | |
WWNPUHZOGTUNGR
|
8.0 | IC50 | 3 | — | |
BGJRUZLMBXELSD
|
8.0 | IC50 | 3 | — | |
BMZFSQDDGKZEHW
|
8.0 | IC50 | 3 | — | |
CAHIWXFAYUQRIN
|
8.0 | IC50 | 2 | — | |
HICLWTCVFGPCRU
|
8.0 | IC50 | 2 | — | |
KLGQSVMIPOVQAX
|
8.0 | IC50 | 7 | — | |
USWRDMVZJWDCCC
|
8.0 | IC50 | 2 | — | |
VKSDILZMXGBZJR
|
8.0 | IC50 | 3 | — | |
WOPOPFZLTYYWDV
|
8.0 | IC50 | 2 | — | |
WQPAUZHGHHSUOT
|
8.0 | IC50 | 3 | — | |
VWKAKGXPHIJGPD
|
8.0 | IC50 | 3 | — | |
JWANSYLSEBELDT
|
7.9 | IC50 | 2 | — | |
NOMOJZWMCUJGHN
|
7.9 | IC50 | 3 | — | |
VERJHOAQBPYQNX
|
7.9 | IC50 | 2 | — | |
AUNVTZZLENFGSL
|
7.9 | IC50 | 2 | — | |
DJNXWSQAIXTYAO
|
7.9 | IC50 | 2 | — | |
FUQQJIVTKMJOTI
|
7.9 | IC50 | 2 | — | |
IRYZTIMDNVDWKI
|
7.9 | IC50 | 2 | — | |
UKLOIUCBRFPROX
|
7.9 | IC50 | 2 | — | |
XWXLFXATFVYHPX
|
7.9 | IC50 | 3 | — | |
ZGHNBPCNVXEKGL
|
7.9 | IC50 | 2 | — | |
ZQAMFUHPGNZLHA
|
7.9 | IC50 | 3 | — | |
HBRPUCMYDQNVOS
|
7.9 | IC50 | 3 | — | |
ARCOJIXZDJYBCH
|
7.9 | IC50 | 2 | — | |
AYRJROJFWRQHPH
|
7.9 | IC50 | 2 | — | |
HJVQHFYHONMFDN
|
7.9 | IC50 | 2 | — | |
QWYIBGOLIBASGM
|
7.9 | IC50 | 2 | — | |
JLVRTMBMCWYGAL
|
7.9 | IC50 | 7 | — | |
CDDNTCUZCTVFFB
|
7.8 | IC50 | 2 | — | |
FZQYCOUBRJEYBC
|
7.8 | IC50 | 2 | — | |
IGUUHDRIMHCZGF
|
7.8 | IC50 | 2 | — | |
RSDNLMODCLIZFE
|
7.8 | IC50 | 2 | — | |
SOUHZJJPQGQXGA
|
7.8 | IC50 | 2 | — | |
TXRJABUPPZKCNT
|
7.8 | IC50 | 2 | — |