Target Details
| UniProt AC | O95271 |
|---|---|
| Gene Symbol | TNKS |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 711
- Clinical molecules 0
- Avg pChEMBL 7.76
Active Molecules (711)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IOYDCKAEKGCUHT
|
8.3 | IC50 | 2 | — | |
QEKJBQMYZARNMZ
|
8.3 | IC50 | 2 | — | |
AONMVAKCMAYUDD
|
8.3 | IC50 | 2 | — | |
BSFWBIWYONWUDM
|
8.3 | IC50 | 2 | — | |
GNQFITKNHVZOAH
|
8.3 | IC50 | 2 | — | |
KVBKYZXBOMQZDK
|
8.3 | IC50 | 2 | — | |
ITFXLHSJWDBGLD
|
8.2 | IC50 | 2 | — | |
VFISXTZNNUCHQR
|
8.2 | IC50 | 2 | — | |
BVCFVQGPDDYTEY
|
8.2 | IC50 | 2 | — | |
PYTOHIUBXSJKQH
|
8.2 | IC50 | 2 | — | |
HKHWXFAGFIXRIT
|
8.2 | IC50 | 2 | — | |
RHCZTJJJLXGIDT
|
8.2 | IC50 | 4 | — | |
ZBQDZIKGERQLAW
|
8.2 | IC50 | 2 | — | |
ACORHZMZJPXEAA
|
8.2 | IC50 | 2 | — | |
MWUSNBQNIIMQRN
|
8.2 | IC50 | 4 | — | |
RLCHCUMPTXYOAE
|
8.2 | IC50 | 2 | — | |
UEPQJCJZMGAYPN
|
8.2 | IC50 | 2 | — | |
UQSSCRPZDDBPIX
|
8.2 | IC50 | 3 | — | |
GWKQMSZYRPKGIR
|
8.2 | IC50 | 3 | — | |
VYNMMNYWFMDPRI
|
8.2 | IC50 | 2 | — | |
YVWYZVHKYSEWDY
|
8.2 | IC50 | 2 | — | |
ASRXCLRFDVRXIO
|
8.2 | IC50 | 2 | — | |
DWXBRPPQEBUSHN
|
8.2 | IC50 | 2 | — | |
AFEVCFCEYWOQKD
|
8.2 | IC50 | 2 | — | |
AXLLIVDKOSPBTM
|
8.2 | IC50 | 3 | — | |
NZVGSVJJAPFBDQ
|
8.2 | IC50 | 2 | — | |
APINASOTMBYJNI
|
8.2 | IC50 | 2 | — | |
GOVCXLYQFHKEOM
|
8.2 | IC50 | 2 | — | |
IZGNMSCICRBUAB
|
8.2 | IC50 | 3 | — | |
YKWFRENASSHRDV
|
8.2 | IC50 | 3 | — | |
BGISDNKMCUOWSJ
|
8.1 | IC50 | 2 | — | |
QCAJKPUKPLDOJH
|
8.1 | IC50 | 2 | — | |
AOHDVRMMHYGYNT
|
8.1 | IC50 | 2 | — | |
PAMGRUFJDHRZSY
|
8.1 | IC50 | 2 | — | |
ZPTIGCVQFHKQDB
|
8.1 | IC50 | 3 | — | |
BCSYLIBZTSVMJI
|
8.1 | IC50 | 3 | — | |
FAANBVRTVUGZKM
|
8.1 | IC50 | 2 | — | |
WSTUZGSSQNKRSR
|
8.1 | IC50 | 2 | — | |
WWKKOAKRYQQEBT
|
8.1 | IC50 | 3 | — | |
MILMCUZGEDRYHA
|
8.1 | IC50 | 3 | — | |
MKFFPXHRRSVHGY
|
8.1 | IC50 | 2 | — | |
OPXFUPAGTLOLPU
|
8.1 | IC50 | 2 | — | |
UXQSFPKVNVQHTR
|
8.1 | IC50 | 2 | — | |
CEKWANGMSIIGAG
|
8.1 | IC50 | 3 | — | |
LLEDTOVGLYBQOU
|
8.1 | IC50 | 2 | — | |
CEPPOYASQJVNOB
|
8.1 | IC50 | 2 | — | |
NHVRXWDQNHZJTK
|
8.1 | IC50 | 3 | — | |
SOHHQHWGZGODEC
|
8.1 | IC50 | 2 | — | |
VUDVJHSDJGLCGJ
|
8.1 | IC50 | 2 | — | |
XMLTXFYPZQGCBX
|
8.1 | IC50 | 2 | — |