Target Details
| UniProt AC | O95271 |
|---|---|
| Gene Symbol | TNKS |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 711
- Clinical molecules 0
- Avg pChEMBL 7.76
Active Molecules (711)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KCXFNUZJEYUGTK
|
8.5 | IC50 | 3 | — | |
AXUQAIVLNXVOPO
|
8.5 | IC50 | 2 | — | |
LDWBPQDBDYNXIG
|
8.5 | IC50 | 2 | — | |
QWYZLCULSMFWLC
|
8.5 | IC50 | 2 | — | |
TUBKWTSXRBZCOP
|
8.5 | IC50 | 2 | — | |
ZRQMVNYALKQFAB
|
8.5 | IC50 | 3 | — | |
YWNDUCFQXOXSHW
|
8.5 | IC50 | 2 | — | |
KOIGSPGBVAOKRC
|
8.5 | IC50 | 2 | — | |
SRAYYDCMTKRHDU
|
8.4 | IC50 | 2 | — | |
VJWOVHIEGPXVQC
|
8.4 | IC50 | 2 | — | |
ZFHIMDPSSCABJV
|
8.4 | IC50 | 2 | — | |
STSCRAGBCYODMY
|
8.4 | IC50 | 8 | — | |
XUAKOEYHACUTGL
|
8.4 | IC50 | 2 | — | |
NKPDQKILCAOJCZ
|
8.4 | IC50 | 2 | — | |
SRMMCJRPCQBABR
|
8.4 | IC50 | 3 | — | |
VJGJUSYNOCTGBZ
|
8.4 | IC50 | 2 | — | |
AANAXNPTHMWCLV
|
8.4 | IC50 | 2 | — | |
DXJNIJJCRJVJHJ
|
8.4 | IC50 | 2 | — | |
FWEQRPGVBGGLAV
|
8.4 | IC50 | 2 | — | |
HOSHPNDTAUJRNF
|
8.4 | IC50 | 2 | — | |
QDVBJHFEZRTDHU
|
8.4 | IC50 | 2 | — | |
RFNNKKMUXMUNHH
|
8.4 | IC50 | 2 | — | |
WADUGMWGTNMWRD
|
8.4 | IC50 | 3 | — | |
ZFSOEIOPMMKKQB
|
8.4 | IC50 | 2 | — | |
CKOUULRCBKAWEI
|
8.4 | IC50 | 4 | — | |
SFJDBLUTKNOEFD
|
8.4 | IC50 | 2 | — | |
OCRURQUHABYGMH
|
8.4 | IC50 | 2 | — | |
VYEHWPWLVNLHOH
|
8.4 | IC50 | 2 | — | |
QHYBVVNCUYAMLN
|
8.4 | IC50 | 2 | — | |
HSKIFVPMPRQUPP
|
8.4 | IC50 | 2 | — | |
OTGSIWARTZTTNU
|
8.4 | IC50 | 2 | — | |
ZBQNBDDBQXSUCN
|
8.4 | IC50 | 2 | — | |
ZHQHQOFGNSFGMK
|
8.4 | IC50 | 2 | — | |
MLYXNNKIUOWZAV
|
8.3 | IC50 | 2 | — | |
VTBFTBOYJMHXBF
|
8.3 | IC50 | 2 | — | |
HJUQWFCFPAEZGB
|
8.3 | IC50 | 2 | — | |
KEKRVUGHUCXWSM
|
8.3 | IC50 | 2 | — | |
KUJBLNYPSGEQPW
|
8.3 | IC50 | 2 | — | |
VNDAUZPOPZSKLR
|
8.3 | IC50 | 2 | — | |
INWWJFRDVLSCGE
|
8.3 | IC50 | 2 | — | |
DGBBDMXUPJSMJV
|
8.3 | IC50 | 2 | — | |
JMPOHTPVCKISQL
|
8.3 | IC50 | 3 | — | |
PQOYFQLZYDRHBS
|
8.3 | IC50 | 2 | — | |
QTABKBZRAZXDQK
|
8.3 | IC50 | 2 | — | |
AQSATLITSNDZSM
|
8.3 | IC50 | 2 | — | |
HBJBOCIRHMWTFT
|
8.3 | IC50 | 3 | — | |
OEHCCJHWIUUHFU
|
8.3 | IC50 | 3 | — | |
VADYPHREEXKWAX
|
8.3 | IC50 | 2 | — | |
YSXKCOVMSIANLW
|
8.3 | IC50 | 2 | — | |
SXGWZNHFZFXRCA
|
8.3 | IC50 | 2 | — |