Target Details
| UniProt AC | O95271 |
|---|---|
| Gene Symbol | TNKS |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 711
- Clinical molecules 0
- Avg pChEMBL 7.76
Active Molecules (711)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CADYSKUZMAIDBU
|
8.9 | IC50 | 4 | — | |
AXAVZUGQTQESKM
|
8.8 | IC50 | 2 | — | |
DYMJRWLCTOEALR
|
8.8 | IC50 | 2 | — | |
GMZHCIWODQRBEX
|
8.8 | IC50 | 2 | — | |
PPGDXAFAEKIBAL
|
8.8 | IC50 | 3 | — | |
PSRZACYIKWDSNE
|
8.8 | IC50 | 2 | — | |
QDFBKHZKWYRNJE
|
8.8 | IC50 | 2 | — | |
TZBJUABBPHUUCL
|
8.8 | IC50 | 3 | — | |
IFGZJOCKQVPMQP
|
8.8 | IC50 | 3 | — | |
IQJONQOJCNHAQX
|
8.8 | IC50 | 2 | — | |
YJZCHZMPLVJNHG
|
8.8 | IC50 | 2 | — | |
FZJXZJRCQJPQDJ
|
8.8 | IC50 | 2 | — | |
QXYNHQXOVDACBV
|
8.8 | IC50 | 2 | — | |
ABCZORPRBCURRK
|
8.8 | IC50 | 3 | — | |
ITIZYYXRCNBXRH
|
8.7 | IC50 | 2 | — | |
JWTZFQHEWRUOBW
|
8.7 | IC50 | 3 | — | |
AOMPHWKJTUPEOB
|
8.7 | IC50 | 3 | — | |
BPRGXQTYABGOBA
|
8.7 | IC50 | 3 | — | |
MGEFDMCHHLACOB
|
8.7 | IC50 | 4 | — | |
ATNQGPSTVULMGA
|
8.7 | IC50 | 2 | — | |
JYHGLYFYVGECPO
|
8.7 | IC50 | 2 | — | |
QTAONPFQLNZKSD
|
8.7 | IC50 | 2 | — | |
UIEGUWBRAAXPAC
|
8.7 | IC50 | 2 | — | |
ZJHLKLRWORVGKO
|
8.7 | IC50 | 3 | — | |
SSRCPYMXFHISQW
|
8.7 | IC50 | 3 | — | |
HEJKSHFADGJFLY
|
8.7 | IC50 | 2 | — | |
OIHAQLWXPNRBJG
|
8.7 | IC50 | 2 | — | |
XTEDLLOZIRDMGM
|
8.7 | IC50 | 3 | — | |
QZHUFUOXNJRYML
|
8.7 | IC50 | 4 | — | |
HIVDAZHBOHYAOK
|
8.6 | IC50 | 2 | — | |
SHCKGNRFHFRCLF
|
8.6 | IC50 | 3 | — | |
VJHDAFXRSRJKPL
|
8.6 | IC50 | 3 | — | |
WQGFJZQGDWKRMN
|
8.6 | IC50 | 4 | — | |
JPLMWQFVSFXHLA
|
8.6 | IC50 | 2 | — | |
ISIFMYDJQDUUNJ
|
8.6 | IC50 | 2 | — | |
JXORYUCIOICGOX
|
8.6 | IC50 | 3 | — | |
KRJJSTRNPUSJST
|
8.6 | IC50 | 2 | — | |
OAXRVCSFISVGCI
|
8.6 | IC50 | 3 | — | |
PBMBCYUKPBTOQE
|
8.6 | IC50 | 2 | — | |
PHWWAZGJHKJDLI
|
8.6 | IC50 | 2 | — | |
XLMMDZKMFSPWBN
|
8.6 | IC50 | 2 | — | |
AOMPHWKJTUPEOB
|
8.6 | IC50 | 3 | — | |
WDAVNQKSHQVPKD
|
8.6 | IC50 | 4 | — | |
BDBCLQYLIMPBKR
|
8.6 | IC50 | 2 | — | |
NLGGKDGPDAYIFS
|
8.5 | IC50 | 2 | — | |
ZJAQFWFBBDESAQ
|
8.5 | IC50 | 3 | — | |
PEOXTCZVHIZAKJ
|
8.5 | IC50 | 2 | — | |
VNRKPTDAMCLGEX
|
8.5 | IC50 | 2 | — | |
WYQKLIGAUQKHIE
|
8.5 | IC50 | 3 | — | |
DPLIWMOJVZZKPZ
|
8.5 | IC50 | 2 | — |