Target Details
| UniProt AC | O95271 |
|---|---|
| Gene Symbol | TNKS |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 711
- Clinical molecules 0
- Avg pChEMBL 7.76
Active Molecules (711)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KCIAHAOBFVPQKW
|
9.3 | IC50 | 2 | — | |
XXNXCOLKURBCKS
|
9.3 | IC50 | 2 | — | |
NUCKGGSDYMOWIS
|
9.3 | IC50 | 2 | — | |
FDICCIFLUUYDFS
|
9.3 | IC50 | 4 | — | |
IGTMNQSNSCDFLH
|
9.3 | IC50 | 2 | — | |
TXRJABUPPZKCNT
|
9.3 | IC50 | 2 | — | |
LPJHLUNKDITEKL
|
9.3 | IC50 | 2 | — | |
AAGQBOZLMIXHHO
|
9.3 | IC50 | 3 | — | |
BTVYOOANNCDQKM
|
9.3 | IC50 | 2 | — | |
ZBYOHASAEQTYGT
|
9.3 | IC50 | 2 | — | |
AICJSAOJHVWPBE
|
9.3 | IC50 | 2 | — | |
NLHWNHOBNJGSMX
|
9.3 | IC50 | 3 | — | |
MONJJZAAKCCXFC
|
9.2 | IC50 | 2 | — | |
CVEOMWCWJJWSAV
|
9.2 | IC50 | 2 | — | |
JCXKRJIIGPWGFB
|
9.2 | IC50 | 2 | — | |
MEQYFMGLIUJKRI
|
9.2 | IC50 | 2 | — | |
ZMDXCCGWVIFDMF
|
9.2 | IC50 | 2 | — | |
MPXAEYSGFKRDQM
|
9.2 | IC50 | 7 | — | |
BGRUEOQGBAKLPG
|
9.2 | IC50 | 2 | — | |
HDYMAMWGPQYCJR
|
9.2 | IC50 | 2 | — | |
QFFQVTQVYJNUQK
|
9.2 | IC50 | 2 | — | |
VQDCXZLOFBIDTL
|
9.2 | IC50 | 2 | — | |
RKTAKASHRFDDHH
|
9.2 | IC50 | 2 | — | |
KTIYJXKGHKLGEV
|
9.2 | IC50 | 3 | — | |
HBWPYEOAXUKSAJ
|
9.2 | IC50 | 2 | — | |
RGSSADMOZOOPCT
|
9.1 | IC50 | 4 | — | |
JDZQHCQYJAHSCQ
|
9.1 | IC50 | 3 | — | |
KCCHUDANIWRWFS
|
9.1 | IC50 | 3 | — | |
PCRNXFSEUXATPP
|
9.1 | IC50 | 2 | — | |
SSRCPYMXFHISQW
|
9.1 | IC50 | 3 | — | |
LMUIMYHRSNNJLB
|
9.1 | IC50 | 2 | — | |
XBMLIULZOSKFDL
|
9.1 | IC50 | 2 | — | |
FUQQJIVTKMJOTI
|
9.1 | IC50 | 2 | — | |
AFHDZWZQZNOEPI
|
9.1 | IC50 | 4 | — | |
OOQHGTMJHBCFLX
|
9.0 | IC50 | 2 | — | |
ANMLHQJBUZSTOM
|
9.0 | IC50 | 2 | — | |
KPDGLOCQRBTKHT
|
9.0 | IC50 | 3 | — | |
UIPJAQKAZCQVPU
|
9.0 | IC50 | 3 | — | |
YFRRHPBZXLBANM
|
9.0 | IC50 | 3 | — | |
FHWNIOZFSDHKSG
|
9.0 | IC50 | 4 | — | |
JKUCQWSEJQYAJC
|
9.0 | IC50 | 3 | — | |
GTRSBOPVOQICBF
|
9.0 | IC50 | 2 | — | |
QKUQIWILQMTNRG
|
9.0 | IC50 | 2 | — | |
ZDXHDNKNNXPLHR
|
9.0 | IC50 | 2 | — | |
JLUWGYRKHZWQDW
|
8.9 | IC50 | 2 | — | |
GWBSSUZALYDTAX
|
8.9 | IC50 | 3 | — | |
OKVSYWJACIIIKC
|
8.9 | IC50 | 2 | — | |
NENMCAZABRSHBQ
|
8.9 | IC50 | 2 | — | |
NRGTYYQXOBIJNO
|
8.9 | IC50 | 3 | — | |
TVAKNHJAERNITR
|
8.9 | IC50 | 2 | — |