Target Details
| UniProt AC | O95271 |
|---|---|
| Gene Symbol | TNKS |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 711
- Clinical molecules 0
- Avg pChEMBL 7.76
Active Molecules (711)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HPVNLHNRECCVHK
|
6.1 | IC50 | 2 | — | |
PPOQMSJVMJCEAI
|
6.1 | IC50 | 2 | — | |
PGAMJHQYVDYIQX
|
6.1 | IC50 | 3 | — | |
NXRCVVIFMJBFPF
|
6.0 | IC50 | 3 | — | |
OFJNKCHKIMIYDT
|
6.0 | IC50 | 2 | — | |
ZXYKQNYSXHNQMV
|
6.0 | IC50 | 6 | — | |
GGQAXNFSEUSJJE
|
6.0 | IC50 | 3 | — | |
KRIKILRRJCIWNB
|
6.0 | IC50 | 5 | — | |
MOYOUBMGSIHZJF
|
6.0 | IC50 | 2 | — | |
OPXUZDOALWXAIC
|
6.0 | IC50 | 2 | — | |
QFWFAXXCERFDCB
|
6.0 | IC50 | 2 | — |