Target Details
| UniProt AC | O95271 |
|---|---|
| Gene Symbol | TNKS |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 711
- Clinical molecules 0
- Avg pChEMBL 7.76
Active Molecules (711)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YFRJWFALOKTWJY
|
6.4 | IC50 | 3 | — | |
ONMIHAIKNBLEMB
|
6.4 | IC50 | 2 | — | |
XMNISQQDQQVTBJ
|
6.4 | IC50 | 4 | — | |
DDFLFKTXUWPNMV
|
6.4 | IC50 | 3 | — | |
DDFLFKTXUWPNMV
|
6.4 | IC50 | 3 | — | |
RDCQUWQHGNCDQF
|
6.4 | IC50 | 3 | — | |
BSGNOJZPCZALIF
|
6.4 | IC50 | 2 | — | |
UYBOMUVIPAWXHH
|
6.4 | IC50 | 2 | — | |
JDCPQGXAZCZLPD
|
6.4 | IC50 | 2 | — | |
LSKQRMBPLLMJRR
|
6.4 | IC50 | 2 | — | |
JXSWEIKYXMJGGG
|
6.3 | IC50 | 3 | — | |
QOUNQNYSBYTMLY
|
6.3 | IC50 | 2 | — | |
WPCRHWQMOWNQPY
|
6.3 | IC50 | 2 | — | |
FMWDCSQWMNXQJI
|
6.3 | IC50 | 2 | — | |
GECCSCOUJAXBHM
|
6.3 | IC50 | 2 | — | |
QNQFPYADHVFRKQ
|
6.3 | IC50 | 5 | — | |
PVRVKAMGYYHFJO
|
6.3 | IC50 | 3 | — | |
YZLWXJLWHXPUGR
|
6.3 | IC50 | 2 | — | |
HMZVOPJPTNTGGO
|
6.3 | IC50 | 2 | — | |
HKKWGEHTJZYRCM
|
6.3 | IC50 | 3 | — | |
NIEJYIGLCXXXQE
|
6.3 | IC50 | 2 | — | |
UAVGSHVHWKPCPP
|
6.3 | IC50 | 3 | — | |
XGSDYBUNVFYCTB
|
6.3 | IC50 | 2 | — | |
ZGSXEXBYLJIOGF
|
6.3 | IC50 | 2 | — | |
BDZQPEDPOGIWQX
|
6.2 | IC50 | 2 | — | |
PFKDFLVWKSDYJO
|
6.2 | IC50 | 2 | — | |
SQVXWIUVAILQRH
|
6.2 | IC50 | 2 | — | |
ZMGPDWHTUMUFPT
|
6.2 | IC50 | 2 | — | |
DUVLGZHVLHPLOD
|
6.2 | IC50 | 2 | — | |
KDEAARCPDWPBIF
|
6.2 | IC50 | 2 | — | |
PCHKPVIQAHNQLW
|
6.2 | IC50 | 8 | — | |
YZHRVEFGEYGJNZ
|
6.2 | IC50 | 2 | — | |
GBJOIXJAQBNTML
|
6.2 | IC50 | 2 | — | |
ZKKFHBDYTOSSFW
|
6.2 | IC50 | 2 | — | |
WXBLUJQGIFPHFK
|
6.2 | IC50 | 3 | — | |
NNQPXWGOYRBSTO
|
6.2 | IC50 | 3 | — | |
CXPJWDXJJXREGA
|
6.2 | IC50 | 3 | — | |
HHQJCXWKFODTFE
|
6.2 | IC50 | 2 | — | |
UKLWMTAVXDIMIA
|
6.2 | IC50 | 2 | — | |
WBYWAXJHAXSJNI
|
6.2 | IC50 | 13 | — | |
WOVOBLGUSQNZJX
|
6.2 | IC50 | 2 | — | |
BVCFVQGPDDYTEY
|
6.2 | IC50 | 2 | — | |
GABWOUPESSRDHY
|
6.2 | IC50 | 2 | — | |
TWBVIDDSIBCAOI
|
6.1 | IC50 | 2 | — | |
IBBZXRLLZKUNIM
|
6.1 | IC50 | 4 | — | |
PHQBXCTZDRMXMX
|
6.1 | IC50 | 2 | — | |
QEFRLEQZTKAQJC
|
6.1 | IC50 | 2 | — | |
SHGLJXBLXNNCTE
|
6.1 | IC50 | 2 | — | |
ZBCTWQCRORRYGT
|
6.1 | IC50 | 2 | — | |
PADREXIRIZBNMQ
|
6.1 | IC50 | 2 | — |