Target Details
| UniProt AC | O95271 |
|---|---|
| Gene Symbol | TNKS |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 711
- Clinical molecules 0
- Avg pChEMBL 7.76
Active Molecules (711)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BLPUCTSDPCUHQQ
|
6.8 | IC50 | 2 | — | |
BMPSOKZAIFFMLK
|
6.8 | IC50 | 6 | — | |
PAMHLAWFGRSETB
|
6.7 | IC50 | 2 | — | |
VDULOAUXSMYUMG
|
6.7 | IC50 | 2 | — | |
KSLHAODJKMKLGY
|
6.7 | IC50 | 2 | — | |
JRDFYUFZPYBDNH
|
6.7 | IC50 | 2 | — | |
FAMOCXKGUZQGHI
|
6.7 | IC50 | 2 | — | |
LQJVOLSLAFIXSV
|
6.7 | IC50 | 4 | — | |
LUYWAGVRXKSNLL
|
6.7 | IC50 | 2 | — | |
BWTOWBOMDHKCDB
|
6.7 | IC50 | 7 | — | |
BPXQHNKTRNOWCL
|
6.7 | IC50 | 2 | — | |
OMOFVXXXQGHNIN
|
6.7 | IC50 | 2 | — | |
QERGZXHGTSDAGX
|
6.7 | IC50 | 2 | — | |
CXANDIUMTJKCEI
|
6.7 | IC50 | 3 | — | |
QOEFYUDGLXWPLV
|
6.7 | IC50 | 2 | — | |
AFXJUCILCGBUNX
|
6.7 | IC50 | 4 | — | |
NXSUDRQGXBEGAK
|
6.7 | IC50 | 2 | — | |
NJBICKNJLHIUBM
|
6.7 | IC50 | 2 | — | |
NRCCYFAMXZIJSC
|
6.7 | IC50 | 3 | — | |
DENYZIUJOTUUNY
|
6.6 | IC50 | 5 | — | |
BUEVXCMRYKDSMY
|
6.6 | IC50 | 2 | — | |
ZWIJUUMFHSAWDX
|
6.6 | IC50 | 3 | — | |
VEVDSJNRSJPWSK
|
6.6 | IC50 | 2 | — | |
QDMLZFDXQMJAJN
|
6.6 | IC50 | 2 | — | |
USJIPGUTADKMST
|
6.6 | IC50 | 2 | — | |
AKHUKZJZNGHOJU
|
6.6 | IC50 | 2 | — | |
IMGVRRFHXDRFEY
|
6.6 | IC50 | 2 | — | |
HVPUASJORDGFQX
|
6.6 | IC50 | 3 | — | |
DUCZLEBAUSAZOC
|
6.6 | IC50 | 2 | — | |
SHHNROIKERFQDX
|
6.6 | IC50 | 2 | — | |
DYARIVMCYYQNNQ
|
6.5 | IC50 | 2 | — | |
KRLQJSZEXYIYPQ
|
6.5 | IC50 | 2 | — | |
TVSSLHKEVCLVAI
|
6.5 | IC50 | 2 | — | |
VRIIEPKACOZIMS
|
6.5 | IC50 | 3 | — | |
GKHVECTULDXARR
|
6.5 | IC50 | 2 | — | |
VNFVQSRTHCEODA
|
6.5 | IC50 | 2 | — | |
WMOFKDNPUXQKFI
|
6.5 | IC50 | 3 | — | |
ISZWRZGKEWQACU
|
6.5 | IC50 | 3 | — | |
QDVBJHFEZRTDHU
|
6.5 | IC50 | 2 | — | |
URZUAHXELZUWFE
|
6.5 | IC50 | 2 | — | |
HWGQMRYQVZSGDQ
|
6.5 | IC50 | 6 | — | |
REUQDXNRIHMJKE
|
6.5 | IC50 | 2 | — | |
VHBFFQKBGNRLFZ
|
6.5 | IC50 | 21 | — | |
OWLIGWULYLQYLA
|
6.5 | IC50 | 2 | — | |
YZNNBKHGBJWVKC
|
6.5 | IC50 | 2 | — | |
LFGACFGWTJMDPZ
|
6.5 | IC50 | 2 | — | |
QUWZBGKVPVWAEZ
|
6.5 | IC50 | 2 | — | |
RWQZTEJSVHLLQJ
|
6.5 | IC50 | 2 | — | |
UTEHUKGJDLVHIH
|
6.5 | IC50 | 3 | — | |
NZSKSXWSNJEOQY
|
6.4 | IC50 | 2 | — |