Target Details
| UniProt AC | O95271 |
|---|---|
| Gene Symbol | TNKS |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 711
- Clinical molecules 0
- Avg pChEMBL 7.76
Active Molecules (711)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VQOYZZRRBUAATK
|
7.0 | IC50 | 2 | — | |
DTMHAFMUJHYVGK
|
7.0 | IC50 | 3 | — | |
SEKWIJSPRHUPBY
|
7.0 | IC50 | 2 | — | |
HFAGPKBDTDCMJD
|
7.0 | IC50 | 2 | — | |
RNMBZYKZMPEIAZ
|
7.0 | IC50 | 2 | — | |
UBRJROSZFSUGRT
|
7.0 | IC50 | 2 | — | |
WCPTUQOMNJBIET
|
7.0 | IC50 | 3 | — | |
JVQZLOAYYRAGPS
|
7.0 | IC50 | 2 | — | |
QDMLZFDXQMJAJN
|
7.0 | IC50 | 2 | — | |
GAIPKACDULOVTC
|
7.0 | IC50 | 3 | — | |
BTCPLJSFXYRLAO
|
7.0 | IC50 | 2 | — | |
IRNPOAKXQQBTOH
|
7.0 | IC50 | 3 | — | |
RZFVLEJOHSLEFR
|
7.0 | IC50 | 4 | — | |
DEGIMKQHUITSSN
|
6.9 | IC50 | 2 | — | |
DIOUPOWEQMDVIF
|
6.9 | IC50 | 2 | — | |
KBJDIRAJFGATGU
|
6.9 | IC50 | 2 | — | |
SPNJDQXXJCQIMB
|
6.9 | IC50 | 2 | — | |
NTQHXNALUQPZJR
|
6.9 | IC50 | 3 | — | |
IPVKOLZRYWATMB
|
6.9 | IC50 | 2 | — | |
LXDLBFDPJLZORZ
|
6.9 | IC50 | 2 | — | |
ZBRBBDJXHBEGHX
|
6.9 | IC50 | 2 | — | |
JXSGDVUWLNGDFI
|
6.9 | IC50 | 3 | — | |
NQNHZFQNGJXOBP
|
6.9 | IC50 | 2 | — | |
ANAQCVXUMUTPJY
|
6.9 | IC50 | 3 | — | |
LCGPTLVHGJYCAG
|
6.9 | IC50 | 2 | — | |
ONWFSNLHAZAPLW
|
6.9 | IC50 | 3 | — | |
UVYVRAATXCFMQQ
|
6.9 | IC50 | 4 | — | |
YMZZEZMOHPNZKY
|
6.9 | IC50 | 2 | — | |
ZGSXEXBYLJIOGF
|
6.9 | IC50 | 2 | — | |
IUHUYCJRJLWYHF
|
6.9 | IC50 | 2 | — | |
GNEZFZTYMMBMNW
|
6.9 | IC50 | 2 | — | |
HYPDQYLAVWCCSO
|
6.8 | IC50 | 2 | — | |
VYTWZXZZBQUQMR
|
6.8 | IC50 | 2 | — | |
HMABYWSNWIZPAG
|
6.8 | IC50 | 12 | — | |
VDQXIGZGRYCKAE
|
6.8 | IC50 | 2 | — | |
ZKUPHCJCVQFXDM
|
6.8 | IC50 | 2 | — | |
NEUUVLLFIFUTLB
|
6.8 | IC50 | 2 | — | |
JKCKQJATUNERKN
|
6.8 | IC50 | 2 | — | |
OGYSABKWWQZOIU
|
6.8 | IC50 | 2 | — | |
IGFHGNCTXXHXTG
|
6.8 | IC50 | 2 | — | |
KZLPIRPQDKFMRG
|
6.8 | IC50 | 3 | — | |
LQPOBZQTJQYWPQ
|
6.8 | IC50 | 2 | — | |
MRRMCZVKSVMVSM
|
6.8 | IC50 | 2 | — | |
OXTYNMCLCNPCJW
|
6.8 | IC50 | 2 | — | |
XZTBVJZEZAGWMB
|
6.8 | IC50 | 3 | — | |
XZVNTIRJCBONRF
|
6.8 | IC50 | 2 | — | |
GODKAOHAYPGVHE
|
6.8 | IC50 | 3 | — | |
OKYYDJHOIYUWSW
|
6.8 | IC50 | 3 | — | |
OGYSABKWWQZOIU
|
6.8 | IC50 | 2 | — | |
ZGSXEXBYLJIOGF
|
6.8 | IC50 | 2 | — |