Target Details
| UniProt AC | O95271 |
|---|---|
| Gene Symbol | TNKS |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 711
- Clinical molecules 0
- Avg pChEMBL 7.76
Active Molecules (711)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FDWCAGLPVGJZGX
|
7.3 | IC50 | 3 | — | |
IZQZQDAOIAJQGM
|
7.3 | IC50 | 2 | — | |
JAQKAGMLMPVHSU
|
7.3 | IC50 | 2 | — | |
JGQITQIJKWQWRA
|
7.3 | IC50 | 3 | — | |
FKPMZNSEGYFIDN
|
7.2 | IC50 | 3 | — | |
HGMPUSYAOCCRQP
|
7.2 | IC50 | 3 | — | |
DGMXWRVMCVATCV
|
7.2 | IC50 | 2 | — | |
UVLMNDHVIKTALN
|
7.2 | IC50 | 2 | — | |
LKAMTFJANBYQPK
|
7.2 | IC50 | 2 | — | |
OMOFVXXXQGHNIN
|
7.2 | IC50 | 2 | — | |
WQQPDDQFWUCFDH
|
7.2 | IC50 | 2 | — | |
ZNLWDFKEMBITLP
|
7.2 | IC50 | 2 | — | |
IAGKBCUKKSAKTF
|
7.2 | IC50 | 3 | — | |
JLLCVKKYSDGUPY
|
7.2 | IC50 | 2 | — | |
CKSVYVHLZNMXLX
|
7.2 | IC50 | 4 | — | |
HXVFMRKSTGSLPO
|
7.2 | IC50 | 2 | — | |
MIQSBYOJTBQSKO
|
7.2 | IC50 | 2 | — | |
NBKVXVGFZZVSGF
|
7.2 | IC50 | 2 | — | |
XNKSDYBDUSFGDT
|
7.2 | IC50 | 2 | — | |
HETSSARHFAGODR
|
7.2 | IC50 | 3 | — | |
ONZUYVRREURPTH
|
7.2 | IC50 | 2 | — | |
PTEZEXVUZXGCLZ
|
7.2 | IC50 | 2 | — | |
RFQQBDRYILMLKX
|
7.2 | IC50 | 2 | — | |
GXCGSCMUTWIBEU
|
7.2 | IC50 | 3 | — | |
YUZGATGNXIWEAT
|
7.2 | IC50 | 2 | — | |
ATLOZOFUVNDOGJ
|
7.1 | IC50 | 2 | — | |
JMPCTCLDKNUTHJ
|
7.1 | IC50 | 4 | — | |
NSJLEHJIFVCZLL
|
7.1 | IC50 | 2 | — | |
PFWLEODBNCMHGH
|
7.1 | IC50 | 3 | — | |
QDPSTTBVXGPQGX
|
7.1 | IC50 | 2 | — | |
VNXUSDDWRYWPQI
|
7.1 | IC50 | 2 | — | |
XYPZDGAOLUTGCF
|
7.1 | IC50 | 2 | — | |
QFPKMPQXSRPUCK
|
7.1 | IC50 | 2 | — | |
CCMLHPSWIFWPCV
|
7.1 | IC50 | 2 | — | |
JBNCQRJFEVFZHX
|
7.1 | IC50 | 2 | — | |
LQZSHPITKSPDLC
|
7.1 | Kd | 2 | — | |
OUWQQYPQZGBQTQ
|
7.1 | IC50 | 2 | — | |
JDRRUNIVJVAXBH
|
7.1 | IC50 | 3 | — | |
FNYTYXJFOSRUTI
|
7.1 | IC50 | 3 | — | |
OAXYPHWHZZNXGF
|
7.1 | IC50 | 2 | — | |
QIPLEHXSZJJEQF
|
7.1 | IC50 | 2 | — | |
HKLQJEGTXNKNIH
|
7.1 | IC50 | 2 | — | |
UYLLGWXNACFQPE
|
7.1 | IC50 | 2 | — | |
JVUGYXTVNFUHII
|
7.0 | IC50 | 2 | — | |
UKEHRENMKMWUKT
|
7.0 | IC50 | 2 | — | |
WFUUHEFQQUZRTP
|
7.0 | IC50 | 2 | — | |
PXMYCATYKFCEDH
|
7.0 | IC50 | 2 | — | |
RLEBLHKNUCJVNF
|
7.0 | IC50 | 2 | — | |
HMWZLZHSWIOIGV
|
7.0 | IC50 | 2 | — | |
JRZCNDNPOQFSAY
|
7.0 | IC50 | 2 | — |