Target Details
| UniProt AC | O95271 |
|---|---|
| Gene Symbol | TNKS |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 711
- Clinical molecules 0
- Avg pChEMBL 7.76
Active Molecules (711)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YDGPFYFZYCIASD
|
7.4 | IC50 | 2 | — | |
YNLLVSRMOMOZDP
|
7.4 | IC50 | 2 | — | |
DKMQJZZVSIJOOY
|
7.4 | IC50 | 2 | — | |
PADREXIRIZBNMQ
|
7.4 | IC50 | 2 | — | |
QSAWMHWYVIPNBM
|
7.4 | IC50 | 2 | — | |
APADCINNEFMGCF
|
7.4 | IC50 | 3 | — | |
PBOOUBWKFXDCRA
|
7.4 | IC50 | 3 | — | |
RXVFAGGDYGCELS
|
7.4 | IC50 | 2 | — | |
SGEGLEFCEAUJJJ
|
7.4 | IC50 | 2 | — | |
UYJZZVDLGDDTCL
|
7.4 | IC50 | 8 | — | |
HPTLPJWLCDNFFX
|
7.4 | IC50 | 2 | — | |
KCPVCFVLESRBRB
|
7.4 | IC50 | 2 | — | |
OQISZWBBYFLJCH
|
7.4 | IC50 | 2 | — | |
HWHBVIKIVWUCPS
|
7.4 | IC50 | 2 | — | |
KGBRRRXNQADTEZ
|
7.4 | IC50 | 2 | — | |
SRVUVWKCPPRJQZ
|
7.4 | IC50 | 2 | — | |
WLZJEOODSSBWMB
|
7.4 | IC50 | 3 | — | |
IKSANVUXVVKHGR
|
7.4 | IC50 | 2 | — | |
KJYQLKOWSQIIBB
|
7.4 | IC50 | 2 | — | |
PADREXIRIZBNMQ
|
7.4 | IC50 | 2 | — | |
QSAWMHWYVIPNBM
|
7.4 | IC50 | 2 | — | |
RKIQHTHWSKPSAF
|
7.4 | IC50 | 2 | — | |
YEMNITGJNFFITC
|
7.4 | IC50 | 2 | — | |
ZMPMZCQDIANEGC
|
7.4 | IC50 | 2 | — | |
ZUBOEZVHUJULCK
|
7.4 | IC50 | 3 | — | |
CCVBOAMGJQRBBT
|
7.3 | IC50 | 3 | — | |
CGRPSBDSLCXTLM
|
7.3 | IC50 | 2 | — | |
CRPORXNANROVBQ
|
7.3 | IC50 | 2 | — | |
HIWVLHPKZNBSBE
|
7.3 | IC50 | 3 | — | |
QOUNQNYSBYTMLY
|
7.3 | IC50 | 2 | — | |
QWKZXCNQEFMJAM
|
7.3 | IC50 | 3 | — | |
XUQMWZKEEWRARY
|
7.3 | IC50 | 2 | — | |
HTWNXILBIKZTTF
|
7.3 | IC50 | 2 | — | |
IFOOEZCGGVWMDI
|
7.3 | IC50 | 3 | — | |
GDPZGQDEZJRADO
|
7.3 | IC50 | 2 | — | |
GNQUPDFWLAMRMB
|
7.3 | IC50 | 2 | — | |
HIWVLHPKZNBSBE
|
7.3 | IC50 | 2 | — | |
BGDLETKJFQIBLX
|
7.3 | IC50 | 2 | — | |
DVRLXVRVRZISDR
|
7.3 | IC50 | 2 | — | |
LZWJZQDOBCFTSD
|
7.3 | IC50 | 2 | — | |
JLFSBHQQXIAQEC
|
7.3 | IC50 | 4 | — | |
NIDNWZWMIAQVNK
|
7.3 | IC50 | 2 | — | |
QONNTUSBURAFST
|
7.3 | IC50 | 4 | — | |
FASROOIKQQJQSJ
|
7.3 | IC50 | 2 | — | |
KFHSJMVNDVHQGS
|
7.3 | IC50 | 2 | — | |
LNBBOOMVYRTUHU
|
7.3 | IC50 | 2 | — | |
NIPIEXNSQBQPML
|
7.3 | IC50 | 2 | — | |
OPHKKQQCOYMLPW
|
7.3 | IC50 | 3 | — | |
ZZCRCAHSCCNAPB
|
7.3 | IC50 | 2 | — | |
UQMFJNOQWLUYIO
|
7.3 | IC50 | 2 | — |