Target Details
| UniProt AC | O95271 |
|---|---|
| Gene Symbol | TNKS |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 711
- Clinical molecules 0
- Avg pChEMBL 7.76
Active Molecules (711)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZTIZYNDBJGONBV
|
10.3 | IC50 | 2 | — | |
ARDLHSGXMZNXNJ
|
10.3 | IC50 | 2 | — | |
YTDAPYITALQSLF
|
10.2 | IC50 | 2 | — | |
RZUVUWOWRCUVFD
|
10.2 | IC50 | 2 | — | |
GEXLAFHLVYHZAG
|
10.1 | IC50 | 2 | — | |
MCMCBDOVNWSRNM
|
10.0 | IC50 | 2 | — | |
MPQCBOWATMYRKR
|
10.0 | IC50 | 2 | — | |
FNCGXYCQTPCQIV
|
10.0 | IC50 | 2 | — | |
IOMJPRIMVDNEHH
|
10.0 | IC50 | 2 | — | |
ORMXFDLXICVSQJ
|
9.9 | IC50 | 2 | — | |
HKIWKJRHIASRSM
|
9.9 | IC50 | 3 | — | |
KKBZHPTWKNTEDP
|
9.9 | IC50 | 2 | — | |
CFKUCYZMLBDUOB
|
9.8 | IC50 | 2 | — | |
PISGRABFIARWBA
|
9.8 | IC50 | 2 | — | |
YKDCXYUWCYJSJW
|
9.8 | IC50 | 2 | — | |
QUTSLYJVINTIIL
|
9.8 | IC50 | 2 | — | |
JUVVMZKFNZPQIT
|
9.8 | IC50 | 3 | — | |
LKLUJAFKWQGZNH
|
9.8 | IC50 | 2 | — | |
VXCLLARJZBLHAR
|
9.8 | IC50 | 2 | — | |
CSZYQIKNQBWYMC
|
9.7 | IC50 | 3 | — | |
DJQNMMNQHCULEE
|
9.7 | IC50 | 2 | — | |
UXHCWVAWIZVATP
|
9.7 | IC50 | 2 | — | |
GMBPALAESNNJFY
|
9.7 | IC50 | 2 | — | |
ZTMJFCMMULUTEL
|
9.7 | IC50 | 2 | — | |
HNNOUHLGNDSYMQ
|
9.7 | IC50 | 2 | — | |
MOMSZDNLTDTPMD
|
9.6 | IC50 | 3 | — | |
MAJDINHMZAHJEQ
|
9.6 | IC50 | 2 | — | |
ZWSDFCUUVVGTIL
|
9.6 | IC50 | 2 | — | |
JWNWTMMYAWEEFL
|
9.6 | IC50 | 2 | — | |
DZBLVRUGYZNTPK
|
9.6 | IC50 | 2 | — | |
XSSGDRWJVHTQAM
|
9.6 | IC50 | 2 | — | |
FGJFFFXLPMJDRZ
|
9.6 | IC50 | 3 | — | |
MAISEOAFNXIHQI
|
9.5 | IC50 | 2 | — | |
SWIOCYMLKFHIEX
|
9.5 | IC50 | 2 | — | |
KTIYJXKGHKLGEV
|
9.5 | IC50 | 3 | — | |
BZWBNQLFSDLENC
|
9.5 | IC50 | 2 | — | |
QXYNHQXOVDACBV
|
9.5 | IC50 | 2 | — | |
ZJNATVSUTRSLJP
|
9.5 | IC50 | 3 | — | |
MKFFPXHRRSVHGY
|
9.5 | IC50 | 3 | — | |
IIMAZMNSHUIJDI
|
9.4 | IC50 | 2 | — | |
JVPFBWSJCYHTIN
|
9.4 | IC50 | 3 | — | |
PPFZSMPPXPFDAK
|
9.4 | IC50 | 2 | — | |
OFLAMXGZJOGJGE
|
9.4 | IC50 | 2 | — | |
RGDWKTYYFMMDGT
|
9.4 | IC50 | 2 | — | |
LBUVXBLWWXNUHN
|
9.4 | IC50 | 2 | — | |
XHNQPDNRQBXYJO
|
9.4 | IC50 | 2 | — | |
YFRRHPBZXLBANM
|
9.4 | IC50 | 2 | — | |
BCSYLIBZTSVMJI
|
9.3 | IC50 | 3 | — | |
MOMSZDNLTDTPMD
|
9.3 | IC50 | 2 | — | |
ANHWOOWZYAWFMI
|
9.3 | IC50 | 2 | — |