Target Details
| UniProt AC | O95267 |
|---|---|
| Gene Symbol | RASGRP1 |
| Protein Name | RAS guanyl-releasing protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00617 (RasGEF) PF00618 (RasGEF_N) |
Summary
- Multi-target molecules 13
- Clinical molecules 0
- Avg pChEMBL 7.88
KEGG Pathways (6)
Associated Diseases (1)
Active Molecules (13)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SIWILCBNYOGJQH
|
9.4 | Ki | 4 | — | |
YHESSERBDSKRDZ
|
9.4 | Ki | 4 | — | |
ZETICKHKBWHSEB
|
9.2 | Ki | 4 | — | |
FKPDQMIETMHJBH
|
9.1 | Ki | 4 | — | |
DDBJOZVQHUZKJJ
|
8.8 | Ki | 4 | — | |
JSXUDEUMWQFINT
|
7.6 | Ki | 3 | — | |
OBNHABKOCPUFDD
|
7.6 | Ki | 3 | — | |
JSXUDEUMWQFINT
|
7.5 | Ki | 3 | — | |
OBNHABKOCPUFDD
|
7.4 | Ki | 3 | — | |
WMOCKUYLGCVFJM
|
7.2 | Ki | 3 | — | |
GNIYOZALILMSSH
|
6.9 | Ki | 3 | — | |
RRGGCASWPGLJTK
|
6.2 | Ki | 3 | — | |
UIOPZRFPFXYNME
|
6.2 | Ki | 3 | — |