Target Details
| UniProt AC | O95263 |
|---|---|
| Gene Symbol | PDE8B |
| Protein Name | High affinity cAMP-specific and IBMX-insensitive 3',5'-cyclic phosphodiesterase 8B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF13426 (PAS_9) PF08629 (PDE8) PF23198 (PDE8A_N) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 16
- Clinical molecules 0
- Avg pChEMBL 8.63
KEGG Pathways (5)
Associated Diseases (3)
Active Molecules (16)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UJLHNYPXKZJKLV
|
10.0 | IC50 | 24 | — | |
KXCOKRBRUWINCT
|
9.9 | IC50 | 24 | — | |
KPFFPWNKWSYQFT
|
9.8 | IC50 | 24 | — | |
GOBQSCBEINUNFL
|
9.6 | IC50 | 24 | — | |
VNLPYEMGHGDRRZ
|
9.5 | IC50 | 2 | — | |
AFCWMWBOATWMJV
|
9.5 | IC50 | 24 | — | |
DKSKKVAOIPURFT
|
9.5 | IC50 | 24 | — | |
BPBDCOLBZYWXHD
|
9.0 | IC50 | 24 | — | |
FMMIDZWTNQYEIY
|
9.0 | IC50 | 24 | — | |
QGTJGTFOISKMAD
|
8.9 | IC50 | 2 | — | |
KTZOPPLFULGANJ
|
8.3 | IC50 | 2 | — | |
DWHZRFMVWCPXSM
|
8.2 | IC50 | 2 | — | |
JTROLECZHRVLFM
|
7.8 | IC50 | 10 | — | |
WZGVFBPGGTVOPK
|
6.6 | IC50 | 2 | — | |
OFZGCAMFVYIIHV
|
6.5 | IC50 | 24 | — | |
JITUOVWOCIXEEZ
|
6.0 | IC50 | 23 | — |