Target Details
| UniProt AC | O95180 |
|---|---|
| Gene Symbol | CACNA1H |
| Protein Name | Voltage-dependent T-type calcium channel subunit alpha-1H |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) |
Summary
- Multi-target molecules 265
- Clinical molecules 0
- Avg pChEMBL 7.14
KEGG Pathways (7)
Associated Diseases (3)
Active Molecules (265)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZOYSXBYVJKWUNQ
|
7.0 | IC50 | 3 | — | |
SIFUDDZFIOEDIJ
|
7.0 | IC50 | 3 | — | |
TYSSPUKARDEYKD
|
7.0 | IC50 | 3 | — | |
RTFHWULQHQDWPK
|
7.0 | IC50 | 26 | — | |
IAUJSDFVZKMDSO
|
7.0 | IC50 | 3 | — | |
PZZIZFJADLSSCF
|
7.0 | IC50 | 3 | — | |
ITXUJDTVHQVSLI
|
7.0 | IC50 | 2 | — | |
FADOETCGECQIPP
|
7.0 | IC50 | 2 | — | |
PDUDKACBOWTICF
|
7.0 | IC50 | 2 | — | |
HCEKERAQUTWNGZ
|
7.0 | IC50 | 2 | — | |
PQGYIWNCWOVQQQ
|
7.0 | IC50 | 3 | — | |
GRKKRAWVMXSXDH
|
6.9 | IC50 | 3 | — | |
HCEKERAQUTWNGZ
|
6.9 | IC50 | 2 | — | |
HOGFUDSYCIPQTO
|
6.8 | IC50 | 3 | — | |
JQAPPDSVWXLUJA
|
6.8 | IC50 | 3 | — | |
WZLIQSYWLDAIOK
|
6.8 | IC50 | 3 | — | |
KUPRRUQAZUUGQL
|
6.8 | IC50 | 2 | — | |
FRFNLRPRBZSCOW
|
6.8 | IC50 | 2 | — | |
BHVVIBWVGOFVIP
|
6.8 | IC50 | 2 | — | |
GLVAZBLDEWPYAU
|
6.8 | IC50 | 2 | — | |
HBNPJJILLOYFJU
|
6.8 | IC50 | 21 | — | |
PJBJXVCGIKTWBK
|
6.8 | IC50 | 2 | — | |
QMZDJOIREVQQSG
|
6.8 | IC50 | 3 | — | |
JXXHRRXILZJBQG
|
6.8 | IC50 | 3 | — | |
WESARZWFBOCZMD
|
6.8 | IC50 | 3 | — | |
YVUQSNJEYSNKRX
|
6.8 | IC50 | 36 | — | |
QKTMLCGPKFUYDS
|
6.8 | IC50 | 2 | — | |
BGWZTGQTWNIEFA
|
6.7 | IC50 | 2 | — | |
YRBFVPQLCITKOD
|
6.7 | IC50 | 2 | — | |
YLBJFQXCNGOXMS
|
6.7 | IC50 | 3 | — | |
WEODGHCRBNDCMW
|
6.7 | IC50 | 3 | — | |
CAFYOFMRFOIFOW
|
6.7 | IC50 | 2 | — | |
DKNXRSVMEGIBRJ
|
6.7 | IC50 | 3 | — | |
FIWDRQDDFFDXFN
|
6.7 | IC50 | 3 | — | |
GERVYTOORWZGGL
|
6.7 | IC50 | 2 | — | |
UXVGOSYIXODHIO
|
6.7 | IC50 | 3 | — | |
DVUQADUMMXGGPJ
|
6.7 | IC50 | 3 | — | |
BGWZTGQTWNIEFA
|
6.7 | IC50 | 2 | — | |
IQLMMMGWBQPWOW
|
6.7 | IC50 | 2 | — | |
UZGLRIDSOPLPQJ
|
6.7 | IC50 | 3 | — | |
SKMGZKUUBGORJW
|
6.7 | IC50 | 3 | — | |
ZHJPLTDABORFRU
|
6.7 | IC50 | 3 | — | |
QGMUDAKKGSLGLA
|
6.6 | IC50 | 3 | — | |
SHBCBFDPLIFTBC
|
6.6 | IC50 | 3 | — | |
QGMUDAKKGSLGLA
|
6.6 | IC50 | 4 | — | |
BUHSWYIQMNHKRJ
|
6.6 | IC50 | 3 | — | |
NCPJBCOUXDTXQP
|
6.6 | IC50 | 3 | — | |
NTXMDWIHQBXDSP
|
6.6 | IC50 | 3 | — | |
PYXDWIWBQXUGPX
|
6.5 | IC50 | 3 | — | |
ZORPYTWLJCWREU
|
6.5 | IC50 | 3 | — |