Target Details
| UniProt AC | O95180 |
|---|---|
| Gene Symbol | CACNA1H |
| Protein Name | Voltage-dependent T-type calcium channel subunit alpha-1H |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) |
Summary
- Multi-target molecules 265
- Clinical molecules 0
- Avg pChEMBL 7.14
KEGG Pathways (7)
Associated Diseases (3)
Active Molecules (265)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TWUDJPWCVJDVTM
|
8.7 | IC50 | 26 | — | |
CQCHOVDIAHVBMQ
|
8.7 | IC50 | 26 | — | |
LQNBSHGSEOTYDZ
|
8.6 | IC50 | 26 | — | |
TYXGRJPOMQEXJV
|
8.5 | IC50 | 26 | — | |
GTVKXVAXHKIMQX
|
8.5 | IC50 | 26 | — | |
QYOBBRSIUQCSCG
|
8.4 | IC50 | 3 | — | |
VYABCIPHYKWXBF
|
8.4 | IC50 | 3 | — | |
INSJIVSXEZBVFI
|
8.3 | IC50 | 3 | — | |
HACCLYCGUNUBJY
|
8.2 | IC50 | 26 | — | |
FRGPFJVINLDQIJ
|
8.2 | IC50 | 26 | — | |
JWDSGJQAZOIVIJ
|
8.2 | IC50 | 3 | — | |
JWZPZXKJEUAZFV
|
8.2 | IC50 | 26 | — | |
VOSFWDZWOGANJL
|
8.2 | IC50 | 3 | — | |
YMZQWRKBOMOMLK
|
8.2 | IC50 | 3 | — | |
WRNOOHMVZMXYDO
|
8.2 | IC50 | 3 | — | |
ATAZIWXKOZRZRN
|
8.2 | IC50 | 3 | — | |
RIAAESBLPRZGAK
|
8.2 | IC50 | 26 | — | |
AJCGCPQKWYQPNQ
|
8.1 | IC50 | 26 | — | |
DAMJJTRLEZYXQM
|
8.1 | IC50 | 26 | — | |
XZPYWTFDULVLJE
|
8.1 | IC50 | 3 | — | |
UXEUCTHNMIENKB
|
8.1 | IC50 | 3 | — | |
QUYJROSEXGBONG
|
8.1 | IC50 | 26 | — | |
IQIKXZMPPBEWAD
|
8.1 | IC50 | 3 | — | |
GQWJSRCPJPOCIP
|
8.1 | IC50 | 3 | — | |
LLMGHFGWQHNRKW
|
8.1 | IC50 | 3 | — | |
OXIUFIQCDNTAED
|
8.1 | IC50 | 26 | — | |
AXNHBUZCZYTXFH
|
8.0 | IC50 | 3 | — | |
YEOAYGDVMJPHGG
|
8.0 | IC50 | 26 | — | |
OSYITGFTDTWGJW
|
8.0 | IC50 | 26 | — | |
FQOZFYKBOBBSJQ
|
8.0 | IC50 | 3 | — | |
CGFZKQYHBPQWQB
|
8.0 | IC50 | 3 | — | |
MPAMSENUCHVPRE
|
8.0 | IC50 | 3 | — | |
UGCISYLUHGKJKT
|
8.0 | IC50 | 26 | — | |
DKIVTKARIWZZCD
|
7.9 | IC50 | 3 | — | |
ODYMRNHTFIFRDV
|
7.9 | IC50 | 3 | — | |
SRGBARMXFGWMTF
|
7.9 | IC50 | 26 | — | |
MXPHMHSONUTZJB
|
7.9 | IC50 | 3 | — | |
SYDUPIQUDQXBIQ
|
7.9 | IC50 | 3 | — | |
CNCRGRBWUATVCP
|
7.8 | IC50 | 26 | — | |
GYBBSOIWVDROMG
|
7.8 | IC50 | 3 | — | |
JDKWHGGZYBTDNT
|
7.8 | IC50 | 3 | — | |
KOKBUUOJONICIJ
|
7.8 | IC50 | 3 | — | |
SHDZUWIULZBHDM
|
7.8 | IC50 | 3 | — | |
YZIYDQGNWSHQSD
|
7.8 | IC50 | 26 | — | |
ZHYCMILLXCWHNK
|
7.8 | IC50 | 3 | — | |
ZMYGBEMRHGJETO
|
7.8 | IC50 | 26 | — | |
IIXYZDSTCZPGGD
|
7.8 | IC50 | 3 | — | |
NOCIOWGNSBLDHC
|
7.8 | IC50 | 26 | — | |
NWSFHJWTWBRJFA
|
7.8 | IC50 | 26 | — | |
YPEYQKOBQFSLNA
|
7.8 | IC50 | 3 | — |