Target Details
| UniProt AC | O95136 |
|---|---|
| Gene Symbol | S1PR2 |
| Protein Name | Sphingosine 1-phosphate receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 90
- Clinical molecules 0
- Avg pChEMBL 7.51
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (90)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LRFKWQGGENFBFO
|
9.1 | IC50 | 5 | — | |
KLULNXUHMWEEKT
|
9.1 | IC50 | 4 | — | |
YIZUZSSLYPDFOC
|
9.1 | IC50 | 4 | — | |
VEAJEWXYGKUGPH
|
9.0 | IC50 | 4 | — | |
JNAQEIPNFVZKSC
|
8.8 | IC50 | 4 | — | |
WTJGTMFQALCKRT
|
8.8 | IC50 | 4 | — | |
PCBMXZQDEQINJG
|
8.8 | IC50 | 4 | — | |
JBPVYJJIRRUCJU
|
8.7 | IC50 | 4 | — | |
VKXANKHCILEVSX
|
8.7 | IC50 | 4 | — | |
FSCOADFARBASQU
|
8.7 | IC50 | 4 | — | |
YFWUAIPFVJAYCH
|
8.7 | IC50 | 4 | — | |
SHISURVONRMBAW
|
8.6 | IC50 | 4 | — | |
SQBXAXYMXPCNON
|
8.5 | IC50 | 4 | — | |
GCTZIVJBMHYJOP
|
8.5 | IC50 | 4 | — | |
DUYSYHSSBDVJSM
|
8.5 | Ki | 5 | — | |
DUYSYHSSBDVJSM
|
8.4 | IC50 | 6 | — | |
KUOMYSKEBPYIAO
|
8.4 | IC50 | 4 | — | |
NSEVTFLGGHULPD
|
8.4 | IC50 | 4 | — | |
XQCABFUJSAESPN
|
8.4 | IC50 | 2 | — | |
NOMBGCXWXBTHTO
|
8.3 | IC50 | 4 | — | |
PGLFYYYVMFEVNN
|
8.3 | IC50 | 4 | — | |
HXDPHSXYLHIVSE
|
8.3 | IC50 | 4 | — | |
LRFKWQGGENFBFO
|
8.2 | IC50 | 5 | — | |
DQXSYKMXKITFAL
|
8.2 | IC50 | 3 | — | |
WFMGEMPWKRJJHM
|
8.2 | IC50 | 3 | — | |
BDZJQGMIIWGSHK
|
8.2 | IC50 | 4 | — | |
REWKMHWDRLICNF
|
8.2 | IC50 | 2 | — | |
GBAYNJCGVHFQTM
|
8.1 | IC50 | 4 | — | |
QTRXSBUIHCYTDW
|
8.0 | IC50 | 2 | — | |
NOMBGCXWXBTHTO
|
8.0 | IC50 | 4 | — | |
PGLFYYYVMFEVNN
|
8.0 | IC50 | 4 | — | |
GOQBSVFOBGVWTA
|
8.0 | IC50 | 2 | — | |
WECRLAZSZWCWDE
|
8.0 | IC50 | 5 | — | |
MAXFFKJVDHGPJO
|
8.0 | IC50 | 2 | — | |
KSAATBXYGYJAQU
|
7.9 | IC50 | 4 | — | |
PGLFYYYVMFEVNN
|
7.9 | IC50 | 4 | — | |
ATXJVJPQVHFGIA
|
7.7 | IC50 | 4 | — | |
BYIXDXLVJKFJLY
|
7.7 | IC50 | 2 | — | |
LPQWCJPFMUGAML
|
7.7 | IC50 | 2 | — | |
LYZKFLGVDKUPAP
|
7.7 | IC50 | 4 | — | |
RNSLRQNDXRSASX
|
7.7 | IC50 | 2 | — | |
AXAGGQQXMQHIFF
|
7.6 | IC50 | 4 | — | |
PGLFYYYVMFEVNN
|
7.6 | IC50 | 4 | — | |
MREVGTRWACILNL
|
7.5 | IC50 | 2 | — | |
MMKMRZFTPGRQEQ
|
7.4 | IC50 | 4 | — | |
BYMIMTPDQNLDHL
|
7.4 | IC50 | 3 | — | |
IYOGKTIRIRHPOH
|
7.4 | IC50 | 6 | — | |
JAMOPMAEOMFXHF
|
7.4 | IC50 | 4 | — | |
NOMBGCXWXBTHTO
|
7.4 | IC50 | 4 | — | |
TWNDWWAUVXKNMU
|
7.3 | IC50 | 4 | — |