Target Details
| UniProt AC | O94925 |
|---|---|
| Gene Symbol | GLS |
| Protein Name | Glutaminase kidney isoform, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12796 (Ank_2) PF17959 (EF-hand_14) PF04960 (Glutaminase) |
Summary
- Multi-target molecules 52
- Clinical molecules 0
- Avg pChEMBL 7.61
KEGG Pathways (9)
Associated Diseases (3)
Active Molecules (52)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HXVUCOSFCZYVMC
|
8.4 | IC50 | 2 | — | |
KRTRGYMEOYWRKI
|
8.4 | IC50 | 2 | — | |
OBPILLODCVCGGI
|
8.3 | IC50 | 2 | — | |
PPNVZFPAEJSAFU
|
8.3 | IC50 | 2 | — | |
VPGRTCFKGYVIOS
|
8.3 | IC50 | 2 | — | |
KOGUOWPXAFIILI
|
8.2 | IC50 | 2 | — | |
TWKLHIDOFDFNQS
|
8.2 | IC50 | 2 | — | |
UGUWNXBXJVUOOD
|
8.2 | IC50 | 2 | — | |
FBMFFBGPUNBCNP
|
8.2 | IC50 | 2 | — | |
HHLUIUZVGQITDO
|
8.2 | IC50 | 2 | — | |
VGPLTIRWBIWICN
|
8.2 | IC50 | 2 | — | |
VUDXDCSKAVJVDG
|
8.2 | IC50 | 2 | — | |
CNASVEIJSMEVSH
|
8.1 | IC50 | 2 | — | |
IKJNBJCYDNHKKV
|
8.1 | IC50 | 2 | — | |
RNBFZCUEZCEVSE
|
8.1 | IC50 | 2 | — | |
ROQOBSHXSCJFAR
|
8.1 | IC50 | 2 | — | |
CWBIRWDPNDFZPG
|
8.1 | IC50 | 2 | — | |
DHMIAMOTWINKLX
|
8.1 | IC50 | 2 | — | |
DVADEAFUNXLALS
|
8.0 | IC50 | 2 | — | |
NMAUBZDNIFLCTD
|
8.0 | IC50 | 2 | — | |
FGMMFWMFTAXXTJ
|
7.9 | IC50 | 2 | — | |
SBUXGYYHDPMLCY
|
7.9 | IC50 | 2 | — | |
VOVSTMPHJJITQQ
|
7.9 | IC50 | 2 | — | |
KNTRXABDMADGSN
|
7.8 | IC50 | 2 | — | |
ZIQOFALFFQRVGP
|
7.8 | IC50 | 2 | — | |
LGBVMKUSZJSCPW
|
7.7 | IC50 | 2 | — | |
OOQPQPACUZLVEV
|
7.7 | IC50 | 2 | — | |
PRAAPINBUWJLGA
|
7.6 | IC50 | 2 | — | |
WUDLRYCRZOUWEQ
|
7.6 | IC50 | 2 | — | |
MBAZZANFKMSLFD
|
7.6 | IC50 | 2 | — | |
HPFHSUDXTMQCGE
|
7.6 | IC50 | 2 | — | |
TWLRNPTTYRKLMF
|
7.5 | IC50 | 2 | — | |
LBUGIVGUIVGPRK
|
7.5 | IC50 | 2 | — | |
YMVAHDWFRWUEDF
|
7.5 | IC50 | 2 | — | |
ZDIISWUXPDGWSE
|
7.5 | IC50 | 2 | — | |
DHPBNOLWZCELSM
|
7.4 | IC50 | 2 | — | |
BBDJFYLWIIYIPJ
|
7.4 | IC50 | 2 | — | |
HHDNNVZKVIMCFG
|
7.3 | IC50 | 2 | — | |
NBONAFZFTXZHGQ
|
7.3 | IC50 | 2 | — | |
ZIPXNTFGVYDBAA
|
7.2 | IC50 | 2 | — | |
ATNJAOBQSYRYGW
|
7.1 | IC50 | 2 | — | |
REFHBOVGIOGXRN
|
7.1 | IC50 | 2 | — | |
IIXRBRRPZFGPJV
|
7.0 | IC50 | 2 | — | |
MDJIPXYRSZHCFS
|
6.9 | IC50 | 2 | — | |
GTBLMEKCKSPWPW
|
6.8 | IC50 | 2 | — | |
ACNUPHZNRLLGPV
|
6.7 | IC50 | 2 | — | |
PUSMTINPXLXYNU
|
6.7 | IC50 | 2 | — | |
PXGKVHIRSKZGDU
|
6.7 | IC50 | 2 | — | |
SXFQBUKKIKMRPM
|
6.6 | IC50 | 2 | — | |
IMZXETXDVAKDSY
|
6.4 | IC50 | 2 | — |