Target Details
| UniProt AC | O94921 |
|---|---|
| Gene Symbol | CDK14 |
| Protein Name | Cyclin-dependent kinase 14 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 90
- Clinical molecules 8
- Avg pChEMBL 7.1
KEGG Pathways (1)
Active Molecules (90)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RDUHJWMAQZUAJC
|
9.4 | IC50 | 2 | — | |
MKEGDIVMNZNFAN
|
8.8 | IC50 | 2 | — | |
TTXFWLWLVPCKRX
|
8.7 | IC50 | 2 | — | |
NMXYXLBBQZYFDW
|
8.6 | IC50 | 4 | — | |
RMCYPGSJEZBAMX
|
8.5 | IC50 | 3 | — | |
NUPTZQFLDCQLOT
|
8.5 | IC50 | 4 | — | |
MANOLJFSBPUXMB
|
8.5 | IC50 | 4 | — | |
JIBHJLIMQZDZRK
|
8.4 | IC50 | 3 | — | |
HGZJEOYIMBIRQI
|
8.2 | IC50 | 4 | — | |
XXFHRRDNOYDSKG
|
8.1 | IC50 | 4 | — | |
RBIXFJAPAZPTDA
|
8.0 | IC50 | 2 | — | |
BQCPUBPCBQLKPP
|
8.0 | IC50 | 3 | — | |
JRNJNYBQQYBCLE
|
8.0 | Kd | 40 | Yes | |
XFCDYHLPKFWDMS
|
8.0 | IC50 | 4 | — | |
HRIOLNMHFYSSLV
|
7.8 | IC50 | 2 | — | |
INKWHXBJAUQYBV
|
7.8 | IC50 | 3 | — | |
NJIDANQIZWLYFH
|
7.8 | IC50 | 4 | — | |
PXQWBBNLJZQDEL
|
7.8 | IC50 | 4 | — | |
OVPNQJVDAFNBDN
|
7.8 | IC50 | 44 | Yes | |
GHOIKFWTAAALKT
|
7.8 | IC50 | 3 | — | |
ODPGGGTTYSGTGO
|
7.8 | Kd | 153 | — | |
YKZGTZJVEPDXGU
|
7.6 | IC50 | 3 | — | |
CXQHYVUVSFXTMY
|
7.5 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
7.5 | Kd | 149 | — | |
PBIJEPSJLJLFIU
|
7.4 | IC50 | 2 | — | |
WLGFXUKKLFKVFW
|
7.4 | IC50 | 2 | — | |
AFFKASZZCVHEBW
|
7.3 | IC50 | 4 | — | |
VODCPWQTCXGQLH
|
7.3 | IC50 | 2 | — | |
FGQPUEPSGPHCAO
|
7.3 | IC50 | 4 | — | |
FZWFQSYPXVHFDQ
|
7.3 | IC50 | 4 | — | |
NJIDANQIZWLYFH
|
7.3 | IC50 | 2 | — | |
XXFHRRDNOYDSKG
|
7.3 | IC50 | 2 | — | |
GFNBVYFIPNPBRU
|
7.2 | IC50 | 2 | — | |
HZPYSAHDRSBARR
|
7.2 | IC50 | 4 | — | |
NBSJZWFDNFWQDN
|
7.2 | IC50 | 29 | — | |
FLAQGMBHZVHXIW
|
7.2 | IC50 | 3 | — | |
RYCOMKGMIRGGDD
|
7.2 | IC50 | 4 | — | |
PNISUJSLRCHJAI
|
7.1 | IC50 | 2 | — | |
OQRVOQIHLQYVLO
|
7.1 | IC50 | 3 | — | |
ZDQOAQIVXDLRDY
|
7.1 | IC50 | 4 | — | |
GSUCKLWXUHHJFW
|
7.1 | IC50 | 2 | — | |
RVKNONNXSNALJV
|
7.1 | IC50 | 21 | — | |
ODWIVHQPIGIBFU
|
7.1 | IC50 | 3 | — | |
FLPXFWJMZVSLBP
|
7.1 | IC50 | 4 | — | |
NHUBHFVMKMFCJA
|
7.1 | IC50 | 2 | — | |
WMORAJAIMFWNGT
|
7.1 | IC50 | 2 | — | |
JXCLUBNKARSPIY
|
7.1 | IC50 | 2 | — | |
RKWGLUFSAMFDLN
|
7.0 | IC50 | 2 | — | |
BIIVYFLTOXDAOV
|
7.0 | Kd | 29 | — | |
BIIVYFLTOXDAOV
|
7.0 | Kd | 82 | Yes |