Target Details
| UniProt AC | O94806 |
|---|---|
| Gene Symbol | PRKD3 |
| Protein Name | Serine/threonine-protein kinase D3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00169 (PH) PF00069 (Pkinase) PF25525 (Ubiquitin_PRKD1_N) |
Summary
- Multi-target molecules 354
- Clinical molecules 117
- Avg pChEMBL 6.89
KEGG Pathways (3)
Active Molecules (354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FTIAKTLRFKSDFR
|
6.1 | Ki | 10 | Yes | |
GHAZVJQMLWOQLP
|
6.1 | Ki | 17 | — | |
IUEBPIPDFMCSTP
|
6.1 | Ki | 29 | — | |
NFMGZVPRGVERNN
|
6.1 | Ki | 44 | — | |
QVNZKVACBBTKSL
|
6.1 | Ki | 38 | — | |
SBFPHSVZEXSHTL
|
6.1 | Ki | 62 | — | |
SGHXFHRRWFLILP
|
6.1 | Ki | 29 | — | |
SHENEEFOURUIBP
|
6.1 | Ki | 29 | — | |
TWCARTFPHQNBPF
|
6.1 | Ki | 16 | — | |
UAQJVFADAYIBGC
|
6.1 | Ki | 23 | — | |
UMYBAQLXZPEUQW
|
6.1 | Ki | 15 | — | |
UTMRCMCLMBDPNW
|
6.1 | Ki | 10 | — | |
VTQQYBGURNVVFE
|
6.1 | Ki | 17 | — | |
WSXYBDKZFNJOTP
|
6.1 | IC50 | 12 | Yes | |
XOVPCPRZRHQFBI
|
6.1 | Ki | 15 | — | |
YGKFZWJWKPZPQM
|
6.1 | Ki | 13 | — | |
YKJSWMAVAKRUAN
|
6.1 | Ki | 19 | — | |
ZPXPEKQMLOAPLT
|
6.1 | Ki | 15 | — | |
MRBNLCLXWRXFJX
|
6.1 | IC50 | 15 | — | |
RYYNGWLOYLRZLK
|
6.1 | Kd | 45 | — | |
GHRBXKFGXPOEGA
|
6.0 | IC50 | 12 | Yes | |
UJIAQDJKSXQLIT
|
6.0 | Kd | 38 | — | |
AKOITYPGORWENQ
|
6.0 | Ki | 2 | — | |
AOBLBPWPSKBHSI
|
6.0 | Ki | 55 | — | |
BPNUQXPIQBZCMR
|
6.0 | Kd | 83 | Yes | |
CSDDCHPGQGWRLI
|
6.0 | Ki | 5 | Yes | |
CXBBWVXSZINRCS
|
6.0 | Ki | 41 | — | |
DBKQWGCVGCVPIP
|
6.0 | Ki | 21 | — | |
DYSRECIVMDGUQU
|
6.0 | Ki | 29 | — | |
FQEODTMNWMDUMD
|
6.0 | Ki | 25 | — | |
GDYZFFBMSBDTAA
|
6.0 | Ki | 60 | — | |
GQGMUKOYILWOIQ
|
6.0 | Ki | 25 | — | |
HZPACYSNLOCDLW
|
6.0 | Ki | 48 | — | |
IJNGXROUMFEKDB
|
6.0 | Ki | 39 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JSDGKSMNPHJDFK
|
6.0 | Ki | 35 | — | |
KGPGFQWBCSZGEL
|
6.0 | Kd | 59 | Yes | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KOZOJNNVQMRVIW
|
6.0 | Ki | 4 | — | |
LNIDFQVRZCDVBI
|
6.0 | Ki | 16 | — | |
LWSORTKUYSYDMP
|
6.0 | IC50 | 12 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MTYMWGNJKDHWGN
|
6.0 | Ki | 18 | — | |
NECQZMQPXFYVOY
|
6.0 | Ki | 26 | — | |
NGOGFTYYXHNFQH
|
6.0 | Ki | 15 | — | |
NKANXQFJJICGDU
|
6.0 | IC50 | 35 | Yes | |
OHPRWVPOPFGLJG
|
6.0 | Ki | 19 | — | |
PTSWSUSIGQQZOO
|
6.0 | Ki | 5 | — | |
QEWSTOOMTBAUAG
|
6.0 | Ki | 17 | — | |
UPYHVTCMTMZKAX
|
6.0 | Ki | 12 | — |