Target Details
| UniProt AC | O94806 |
|---|---|
| Gene Symbol | PRKD3 |
| Protein Name | Serine/threonine-protein kinase D3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00169 (PH) PF00069 (Pkinase) PF25525 (Ubiquitin_PRKD1_N) |
Summary
- Multi-target molecules 354
- Clinical molecules 117
- Avg pChEMBL 6.89
KEGG Pathways (3)
Active Molecules (354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DZGATJHVQUFYSK
|
6.3 | Ki | 12 | — | |
HEKAIDKUDLCBRU
|
6.3 | Ki | 20 | — | |
ICDHVAJOGIGIOI
|
6.3 | Ki | 5 | — | |
LRESELHEXSUQGE
|
6.3 | Ki | 10 | — | |
LSLPDHNUWRDOGC
|
6.3 | Ki | 25 | — | |
OADRBDVURCEKRP
|
6.3 | Ki | 44 | — | |
SMRWVXLSRJWVBF
|
6.3 | Ki | 25 | — | |
SPYHMOFSJGTUNP
|
6.3 | Ki | 9 | — | |
UJBJWYNPUOLFIZ
|
6.3 | Ki | 49 | — | |
UVZVWLFSZNPMBS
|
6.3 | Ki | 17 | — | |
VSVWQTDDGQSGHP
|
6.3 | Ki | 51 | — | |
WIHAOLDOGQOGIU
|
6.3 | Ki | 5 | — | |
XKFTZKGMDDZMJI
|
6.3 | Ki | 56 | — | |
KTEIFNKAUNYNJU
|
6.3 | Kd | 114 | — | |
JSPAUBUYPPZXSG
|
6.3 | Ki | 17 | Yes | |
ORNADCNXUPZOQN
|
6.3 | IC50 | 15 | — | |
LOLPPWBBNUVNQZ
|
6.3 | Kd | 97 | Yes | |
NEGCBIBMPAHBIM
|
6.3 | IC50 | 12 | Yes | |
BAQFZMFDZMQJAM
|
6.2 | IC50 | 12 | Yes | |
VXBAJLGYBMTJCY
|
6.2 | Kd | 34 | Yes | |
TXBFOGDMTCNBBT
|
6.2 | IC50 | 12 | Yes | |
QQKKPWJFHBFCTH
|
6.2 | IC50 | 10 | Yes | |
TWUWFRLZDWDJLT
|
6.2 | Ki | 10 | Yes | |
ZUKHVOLIPVGCHQ
|
6.2 | Ki | 10 | Yes | |
GDQXJQSQYMMKRA
|
6.2 | IC50 | 15 | — | |
ZECOHPFWGOCWLO
|
6.2 | IC50 | 5 | — | |
HLXIFVDYTGEUJV
|
6.2 | IC50 | 15 | Yes | |
IILNBGZKSQQREW
|
6.2 | Ki | 6 | — | |
JCFJQIHDZHHMQT
|
6.2 | Ki | 42 | — | |
PAIFYAZSILXLBO
|
6.2 | Ki | 26 | — | |
PHWHNHYZZNJPLB
|
6.2 | Ki | 16 | — | |
PROLIXHVRCJEFH
|
6.2 | Ki | 46 | — | |
QKFXSCNWJZKJSJ
|
6.2 | Ki | 7 | — | |
RIBBPSYZBQQTQC
|
6.2 | Ki | 15 | — | |
UDFDIIVNIYWXDM
|
6.2 | Ki | 74 | — | |
VOAZYSSSBBQYMU
|
6.2 | Ki | 4 | — | |
YMSZHISTTIUBDG
|
6.2 | Ki | 7 | — | |
ZKHDDJKHTPLPOQ
|
6.2 | Ki | 62 | — | |
ZLVOTRRGLSDLPF
|
6.2 | Ki | 36 | — | |
KPJDEGAKXAUVAC
|
6.2 | Ki | 15 | Yes | |
XZXHXSATPCNXJR
|
6.2 | Kd | 165 | Yes | |
CWFIQHQECWPWQG
|
6.2 | IC50 | 16 | Yes | |
ORNADCNXUPZOQN
|
6.2 | IC50 | 15 | — | |
XQJWTJLJEYIUDZ
|
6.2 | IC50 | 2 | — | |
AXTAPYRUEKNRBA
|
6.1 | IC50 | 24 | — | |
JTVBXQAYBIJXRP
|
6.1 | Kd | 20 | — | |
OUSFTKFNBAZUKL
|
6.1 | Kd | 58 | Yes | |
YYLKKYCXAOBSRM
|
6.1 | Kd | 191 | — | |
CPGKMMMSMJKHDL
|
6.1 | Ki | 16 | — | |
DKXHSOUZPMHNIZ
|
6.1 | Ki | 51 | Yes |