Target Details
| UniProt AC | O94806 |
|---|---|
| Gene Symbol | PRKD3 |
| Protein Name | Serine/threonine-protein kinase D3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00169 (PH) PF00069 (Pkinase) PF25525 (Ubiquitin_PRKD1_N) |
Summary
- Multi-target molecules 354
- Clinical molecules 117
- Avg pChEMBL 6.89
KEGG Pathways (3)
Active Molecules (354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AYCPARAPKDAOEN
|
6.6 | Kd | 73 | — | |
IXOVKVHWGKDXKQ
|
6.6 | IC50 | 12 | Yes | |
BRZYOTMFHLERHD
|
6.5 | Ki | 17 | Yes | |
NJEBVFDXJAFAGB
|
6.5 | IC50 | 3 | — | |
WINHZLLDWRZWRT
|
6.5 | Kd | 201 | Yes | |
XLSYZSRXVVCHLS
|
6.5 | Kd | 48 | — | |
XNKIVXYFRPYKHO
|
6.5 | IC50 | 12 | Yes | |
BIIVYFLTOXDAOV
|
6.5 | Ki | 31 | — | |
FLEAYYMORDPWAJ
|
6.5 | Ki | 90 | — | |
KAKGFGCTONHQJW
|
6.5 | Ki | 25 | — | |
MCKPYPWHBUXLEZ
|
6.5 | Ki | 21 | — | |
TVIALAOHRQNPOI
|
6.5 | IC50 | 12 | Yes | |
UCOWZARZLHNDKP
|
6.5 | Ki | 8 | — | |
UYJNQQDJUOUFQJ
|
6.5 | Ki | 68 | — | |
XJJYJNMNYDNXNO
|
6.5 | Ki | 23 | — | |
XXSPHNFKLDJDAK
|
6.5 | Ki | 26 | — | |
GGFLGGNNYKCRAV
|
6.5 | IC50 | 3 | — | |
HPCPUHOULFPBCQ
|
6.5 | IC50 | 12 | Yes | |
JDZXLEPJWLCESI
|
6.5 | IC50 | 12 | Yes | |
RHBWAFDCVFMIFK
|
6.5 | IC50 | 12 | Yes | |
XQVVPGYIWAGRNI
|
6.5 | Kd | 34 | — | |
KTEIFNKAUNYNJU
|
6.5 | Ki | 48 | — | |
RPLXVENRWORMRX
|
6.4 | IC50 | 12 | Yes | |
BMGQWWVMWDBQGC
|
6.4 | IC50 | 147 | Yes | |
MQFYZWYYZGTHAN
|
6.4 | IC50 | 14 | — | |
AHJRHEGDXFFMBM
|
6.4 | Ki | 28 | — | |
DFMCXVONDDGQIY
|
6.4 | Ki | 66 | — | |
DWTNLZZEPSCAIH
|
6.4 | Ki | 25 | — | |
HHLKZSJXDAZIGG
|
6.4 | IC50 | 10 | Yes | |
HSMUWLLZAZCLHF
|
6.4 | Ki | 25 | — | |
LRZYYIZFBXFSJB
|
6.4 | Ki | 69 | — | |
MHWHPWMWKYXCRJ
|
6.4 | Ki | 32 | — | |
NOBMKUVHFRVBES
|
6.4 | Ki | 19 | — | |
SKKRZILJUKYLJS
|
6.4 | Ki | 25 | — | |
UGUZOLHBLLTLBA
|
6.4 | Ki | 15 | — | |
UIRCQOKSJDLYBB
|
6.4 | Ki | 50 | — | |
UQNNJYLAPYGZBD
|
6.4 | Ki | 28 | — | |
WHVFDYQCAMPLMS
|
6.4 | Ki | 20 | Yes | |
WZISGNDZZPSYRP
|
6.4 | Ki | 20 | — | |
ZGDYBJXDIXVTLV
|
6.4 | Ki | 54 | — | |
HZTYDQRUAWIZRE
|
6.4 | Kd | 40 | Yes | |
KAJXOWFGKYKMMZ
|
6.4 | IC50 | 26 | Yes | |
ZFNQOYBHHLGQDV
|
6.3 | IC50 | 12 | Yes | |
HZCVZGCAUBUBST
|
6.3 | IC50 | 3 | — | |
BMBIKZHGTPMMMM
|
6.3 | IC50 | 14 | — | |
CPRVBHBRBVVLHL
|
6.3 | IC50 | 11 | — | |
GUBJNPWVIUFSTR
|
6.3 | Kd | 103 | — | |
CSGQVNMSRKWUSH
|
6.3 | Kd | 21 | — | |
ATBAETXFFCOZOY
|
6.3 | IC50 | 39 | — | |
CCRCRSXDKXZDGK
|
6.3 | IC50 | 12 | Yes |