Target Details
| UniProt AC | O94806 |
|---|---|
| Gene Symbol | PRKD3 |
| Protein Name | Serine/threonine-protein kinase D3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00169 (PH) PF00069 (Pkinase) PF25525 (Ubiquitin_PRKD1_N) |
Summary
- Multi-target molecules 354
- Clinical molecules 117
- Avg pChEMBL 6.89
KEGG Pathways (3)
Active Molecules (354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KXPWWMPXNUOYOH
|
6.8 | Ki | 24 | — | |
NVINUNQBDNEMSY
|
6.8 | Ki | 4 | — | |
OOPMDKIRVTXOPT
|
6.8 | IC50 | 11 | — | |
ORUUEFDGYYTXAF
|
6.8 | Ki | 26 | — | |
OUJZYQBEFNDJQN
|
6.8 | Ki | 71 | — | |
WVFWTUJEHMVUBG
|
6.8 | Ki | 25 | — | |
XFWUTMHVDGPWLH
|
6.8 | Ki | 75 | — | |
BIIVYFLTOXDAOV
|
6.8 | Kd | 29 | — | |
BIIVYFLTOXDAOV
|
6.8 | Kd | 82 | Yes | |
JCHWETQOLSPUBV
|
6.8 | IC50 | 14 | — | |
JHKZENPNLYAVCT
|
6.8 | IC50 | 15 | Yes | |
VWVYILCFSYNJHF
|
6.8 | IC50 | 49 | — | |
OQSTWXKHTZWKLD
|
6.8 | IC50 | 15 | Yes | |
XBAIEEJJCJHBDL
|
6.8 | Ki | 17 | — | |
DQYBRTASHMYDJG
|
6.7 | IC50 | 13 | Yes | |
LGSHHKIOBFPSEK
|
6.7 | IC50 | 12 | Yes | |
BOJKFRKNLSCGHY
|
6.7 | Ki | 10 | Yes | |
DQPYZHUAILXFJI
|
6.7 | Ki | 27 | — | |
FDVSOQRNTAPCHB
|
6.7 | Ki | 40 | — | |
FGWOKLCRQJXPPQ
|
6.7 | Ki | 14 | — | |
GQLWKGVBOIYMTN
|
6.7 | Ki | 35 | — | |
HHSVICUMCOBRPT
|
6.7 | Ki | 33 | — | |
JJJSCYSPSKBQAX
|
6.7 | Ki | 34 | — | |
LHQWPYOYDRVMFI
|
6.7 | Ki | 21 | — | |
MGNQNQOSSLCUFP
|
6.7 | Ki | 12 | — | |
RGNHKJWHFIPHIM
|
6.7 | Ki | 66 | — | |
TVUWQDLBEOZVOU
|
6.7 | Ki | 41 | — | |
TWUWFRLZDWDJLT
|
6.7 | Ki | 10 | Yes | |
XNEPVLVYFUGJLF
|
6.7 | Ki | 27 | — | |
NTXWXFSAJRMWNA
|
6.7 | IC50 | 15 | — | |
RAOJISQDGOOXTK
|
6.7 | IC50 | 14 | Yes | |
MEXUTNIFSHFQRG
|
6.7 | IC50 | 21 | Yes | |
GZJKVFKNTQXSQM
|
6.7 | IC50 | 12 | Yes | |
ZHMXXVNQAFCXKK
|
6.7 | IC50 | 15 | — | |
AACFPJSJOWQNBN
|
6.6 | IC50 | 4 | — | |
MZNUNTIEUOYNNT
|
6.6 | IC50 | 12 | Yes | |
OXEOHAXVZADDOC
|
6.6 | IC50 | 12 | Yes | |
YSVVBGPTTSJYPA
|
6.6 | IC50 | 12 | Yes | |
KOZFSFOOLUUIGY
|
6.6 | IC50 | 26 | — | |
LACOMQAWPSFXQC
|
6.6 | Ki | 27 | — | |
NVRXTLZYXZNATH
|
6.6 | Ki | 47 | Yes | |
ODNOTLMFNVWFTJ
|
6.6 | Ki | 11 | — | |
OWFLADWRSCINST
|
6.6 | Ki | 30 | — | |
QMGUOJYZJKLOLH
|
6.6 | IC50 | 21 | Yes | |
SRONQUHCRFZABC
|
6.6 | Ki | 28 | — | |
SSZFVGXDYBMVDD
|
6.6 | IC50 | 12 | Yes | |
URNZTLZSAVLTIZ
|
6.6 | Ki | 26 | — | |
VSPFURGQAYMVAN
|
6.6 | Ki | 17 | — | |
PBCZSGKMGDDXIJ
|
6.6 | IC50 | 12 | Yes | |
LAOIBIIMKUINJL
|
6.6 | IC50 | 12 | Yes |