Target Details
| UniProt AC | O94806 |
|---|---|
| Gene Symbol | PRKD3 |
| Protein Name | Serine/threonine-protein kinase D3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00169 (PH) PF00069 (Pkinase) PF25525 (Ubiquitin_PRKD1_N) |
Summary
- Multi-target molecules 354
- Clinical molecules 117
- Avg pChEMBL 6.89
KEGG Pathways (3)
Active Molecules (354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZCCPLJOKGAACRT
|
7.1 | Kd | 599 | — | |
CEWOYNHYISZPFC
|
7.1 | IC50 | 3 | — | |
GRENHRYHWHSBLM
|
7.1 | IC50 | 12 | Yes | |
WHROQBPMBHWWTB
|
7.1 | IC50 | 3 | — | |
JZTOUVBEZONDKA
|
7.1 | Ki | 80 | — | |
LCHCSKHPVCDXAU
|
7.1 | Ki | 30 | — | |
LGCKGDRUTNACTA
|
7.1 | IC50 | 11 | — | |
OFPFIAWWDTYSBZ
|
7.1 | Ki | 15 | Yes | |
QAJPIJHWTGPUNZ
|
7.1 | Ki | 37 | — | |
RFBPWKMQWSIPEO
|
7.1 | Ki | 28 | — | |
RHLRPKGACJKWPF
|
7.1 | IC50 | 12 | Yes | |
RYYNGWLOYLRZLK
|
7.1 | Ki | 104 | — | |
VNDWQCSOSCCWIP
|
7.1 | Ki | 39 | Yes | |
XPHWIERLJBFPFV
|
7.1 | Ki | 69 | — | |
GGQAEINRBKFRGZ
|
7.1 | IC50 | 15 | Yes | |
NHDDTLMPCVOXFH
|
7.1 | IC50 | 16 | Yes | |
QQWUGDVOUVUTOY
|
7.0 | Kd | 231 | Yes | |
XDJCLCLBSGGNKS
|
7.0 | Kd | 21 | — | |
FWXIKQAZCDAIKV
|
7.0 | IC50 | 3 | — | |
DKZYXHCYPUVGAF
|
7.0 | Kd | 112 | — | |
SXDPQGRNHSLZPC
|
7.0 | IC50 | 18 | — | |
AILRADAXUVEEIR
|
7.0 | IC50 | 75 | — | |
MQCCJEYZKWZQHU
|
7.0 | IC50 | 15 | Yes | |
YSVVBGPTTSJYPA
|
7.0 | IC50 | 13 | Yes | |
KGMSYXGSYGEHIS
|
7.0 | IC50 | 4 | — | |
KRIUNPBAQZGFQA
|
7.0 | Ki | 76 | — | |
LYNBNVBMAGDJRW
|
7.0 | Ki | 81 | — | |
PFAZIMNYEBJHOA
|
7.0 | IC50 | 12 | Yes | |
UYGYYOIUVFMGKQ
|
7.0 | Ki | 30 | — | |
XRFOMFNAMTYCFF
|
7.0 | IC50 | 12 | Yes | |
YUAWUNMKPARPJD
|
7.0 | IC50 | 14 | Yes | |
BERLXWPRSBJFHO
|
7.0 | IC50 | 4 | — | |
XSHQBIXMLULFEV
|
7.0 | IC50 | 13 | — | |
RBZLXANOQRQGTN
|
7.0 | IC50 | 3 | — | |
KOZFSFOOLUUIGY
|
6.9 | IC50 | 15 | Yes | |
BFSMGDJOXZAERB
|
6.9 | Kd | 33 | — | |
DLWMVUDMPMKGEE
|
6.9 | Ki | 24 | — | |
OGJTZCZJWZSZBT
|
6.9 | IC50 | 12 | Yes | |
WYOMXSAYYXBPMN
|
6.9 | Ki | 24 | — | |
XQVVPGYIWAGRNI
|
6.9 | Ki | 19 | — | |
XYZNKCSDQRKAFR
|
6.9 | Ki | 53 | — | |
ZYTFPHRVOZXPGZ
|
6.9 | Ki | 30 | — | |
VWHZWDRIMLETBG
|
6.9 | IC50 | 12 | Yes | |
DRCBMJUPXHWGMN
|
6.8 | IC50 | 15 | Yes | |
JWVXPOMGWPAEAJ
|
6.8 | IC50 | 10 | Yes | |
QNULKTUETCUJKC
|
6.8 | IC50 | 14 | Yes | |
CZIVUSJISIAXJB
|
6.8 | IC50 | 18 | — | |
BPNUQXPIQBZCMR
|
6.8 | Ki | 60 | — | |
CKVWQORGCCEYHS
|
6.8 | Ki | 50 | — | |
HOYRWTWZUFFACV
|
6.8 | Ki | 28 | — |