Target Details
UniProt ACO94806
Gene SymbolPRKD3
Protein NameSerine/threonine-protein kinase D3
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00130 (C1_1) PF00169 (PH) PF00069 (Pkinase) PF25525 (Ubiquitin_PRKD1_N)
Summary
  • Multi-target molecules 354
  • Clinical molecules 117
  • Avg pChEMBL 6.89
Top Co-occurrence Targets
Active Molecules (354)
InChIKey pChEMBL Type Targets Clinical
PBCZSGKMGDDXIJ 7.8 IC50 68 Yes
XUFLBSMTYMFOQH 7.8 Ki 43
YMIJUBCSOKSFRU 7.8 Ki 87
GTWNYADDKACXSW 7.8 IC50 3
LSEXYAQECWMUPY 7.8 IC50 3
FXGHOAZJQNLNFD 7.8 IC50 13 Yes
HKSZLNNOFSGOKW 7.7 Kd 213
AZIMEXGKUWHPQV 7.7 IC50 12 Yes
CLRFYTGANQZOBS 7.7 Ki 41
FSBMWCWKNXQVMP 7.7 IC50 12 Yes
MZIOLOXGGOLJMJ 7.7 Ki 12
YUKJJLKBBAFYNN 7.7 IC50 12 Yes
KPCVAMMFCPIUIU 7.5 IC50 12 Yes
XXDWSQPJTJZKSJ 7.5 IC50 12 Yes
ZZSBPGIGIUFJRA 7.5 IC50 15 Yes
FELQRVDTGNDOSI 7.5 IC50 15 Yes
JWQOJVOKBAAAAR 7.5 Ki 29
MVJMMLFMPWITEJ 7.5 Ki 110
MYOUXQLHWTWXON 7.5 IC50 16 Yes
PLHUMPJXRHMFFR 7.5 Ki 28
VXYDJXMHISGSDA 7.5 Ki 59
YDZJEODKNRAYMA 7.5 IC50 12 Yes
ZYUGNHPOVKADFZ 7.5 IC50 11
HPBJQOWLAKYNDM 7.4 IC50 15 Yes
AMSOPBXQXSAAAC 7.4 IC50 12 Yes
KOZFSFOOLUUIGY 7.4 IC50 88 Yes
HKSZLNNOFSGOKW 7.4 Ki 118
KJGUOQMSLKZPAT 7.4 IC50 17 Yes
OWRXHGAFWZFFCW 7.4 Ki 113
NTUVEMUMVHHACY 7.4 IC50 12 Yes
AWJAAKKEYXUCFY 7.4 IC50 5
WKZTVBCDQYBGBO 7.3 IC50 16 Yes
AKWVKIGCMCHYJT 7.3 Ki 8
BGYVWFZMYBWCNY 7.3 Ki 30
BMGQWWVMWDBQGC 7.3 IC50 91 Yes
KTWBYGUSEYSRND 7.3 Ki 28
MDHNNGDJYHAYKJ 7.3 IC50 12 Yes
DHUAGGSHTKPOHU 7.3 IC50 3
ZUYALLZMSFUHFE 7.2 IC50 3
XXIWRTOLXWAEJC 7.2 IC50 13 Yes
ACSYKUPGCXYRRO 7.2 Ki 26
DTMZXHDQZQLTHA 7.2 Ki 21
IFPPYSWJNWHOLQ 7.2 Ki 52 Yes
PCQMERRARZKTPW 7.2 Ki 68
RKUKAACYUCUJEE 7.2 Ki 58
TUBBFDZWFNUZLH 7.2 IC50 12 Yes
YEHCNYAQEBQCCS 7.2 Ki 74
HUXYBQXJVXOMKX 7.2 Kd 28
NRUVICOXXLOXCB 7.2 IC50 13 Yes
MGMNDPRNDCWSMZ 7.2 IC50 12 Yes
2D structure