Target Details
| UniProt AC | O94806 |
|---|---|
| Gene Symbol | PRKD3 |
| Protein Name | Serine/threonine-protein kinase D3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00169 (PH) PF00069 (Pkinase) PF25525 (Ubiquitin_PRKD1_N) |
Summary
- Multi-target molecules 354
- Clinical molecules 117
- Avg pChEMBL 6.89
KEGG Pathways (3)
Active Molecules (354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PBCZSGKMGDDXIJ
|
7.8 | IC50 | 68 | Yes | |
XUFLBSMTYMFOQH
|
7.8 | Ki | 43 | — | |
YMIJUBCSOKSFRU
|
7.8 | Ki | 87 | — | |
GTWNYADDKACXSW
|
7.8 | IC50 | 3 | — | |
LSEXYAQECWMUPY
|
7.8 | IC50 | 3 | — | |
FXGHOAZJQNLNFD
|
7.8 | IC50 | 13 | Yes | |
HKSZLNNOFSGOKW
|
7.7 | Kd | 213 | — | |
AZIMEXGKUWHPQV
|
7.7 | IC50 | 12 | Yes | |
CLRFYTGANQZOBS
|
7.7 | Ki | 41 | — | |
FSBMWCWKNXQVMP
|
7.7 | IC50 | 12 | Yes | |
MZIOLOXGGOLJMJ
|
7.7 | Ki | 12 | — | |
YUKJJLKBBAFYNN
|
7.7 | IC50 | 12 | Yes | |
KPCVAMMFCPIUIU
|
7.5 | IC50 | 12 | Yes | |
XXDWSQPJTJZKSJ
|
7.5 | IC50 | 12 | Yes | |
ZZSBPGIGIUFJRA
|
7.5 | IC50 | 15 | Yes | |
FELQRVDTGNDOSI
|
7.5 | IC50 | 15 | Yes | |
JWQOJVOKBAAAAR
|
7.5 | Ki | 29 | — | |
MVJMMLFMPWITEJ
|
7.5 | Ki | 110 | — | |
MYOUXQLHWTWXON
|
7.5 | IC50 | 16 | Yes | |
PLHUMPJXRHMFFR
|
7.5 | Ki | 28 | — | |
VXYDJXMHISGSDA
|
7.5 | Ki | 59 | — | |
YDZJEODKNRAYMA
|
7.5 | IC50 | 12 | Yes | |
ZYUGNHPOVKADFZ
|
7.5 | IC50 | 11 | — | |
HPBJQOWLAKYNDM
|
7.4 | IC50 | 15 | Yes | |
AMSOPBXQXSAAAC
|
7.4 | IC50 | 12 | Yes | |
KOZFSFOOLUUIGY
|
7.4 | IC50 | 88 | Yes | |
HKSZLNNOFSGOKW
|
7.4 | Ki | 118 | — | |
KJGUOQMSLKZPAT
|
7.4 | IC50 | 17 | Yes | |
OWRXHGAFWZFFCW
|
7.4 | Ki | 113 | — | |
NTUVEMUMVHHACY
|
7.4 | IC50 | 12 | Yes | |
AWJAAKKEYXUCFY
|
7.4 | IC50 | 5 | — | |
WKZTVBCDQYBGBO
|
7.3 | IC50 | 16 | Yes | |
AKWVKIGCMCHYJT
|
7.3 | Ki | 8 | — | |
BGYVWFZMYBWCNY
|
7.3 | Ki | 30 | — | |
BMGQWWVMWDBQGC
|
7.3 | IC50 | 91 | Yes | |
KTWBYGUSEYSRND
|
7.3 | Ki | 28 | — | |
MDHNNGDJYHAYKJ
|
7.3 | IC50 | 12 | Yes | |
DHUAGGSHTKPOHU
|
7.3 | IC50 | 3 | — | |
ZUYALLZMSFUHFE
|
7.2 | IC50 | 3 | — | |
XXIWRTOLXWAEJC
|
7.2 | IC50 | 13 | Yes | |
ACSYKUPGCXYRRO
|
7.2 | Ki | 26 | — | |
DTMZXHDQZQLTHA
|
7.2 | Ki | 21 | — | |
IFPPYSWJNWHOLQ
|
7.2 | Ki | 52 | Yes | |
PCQMERRARZKTPW
|
7.2 | Ki | 68 | — | |
RKUKAACYUCUJEE
|
7.2 | Ki | 58 | — | |
TUBBFDZWFNUZLH
|
7.2 | IC50 | 12 | Yes | |
YEHCNYAQEBQCCS
|
7.2 | Ki | 74 | — | |
HUXYBQXJVXOMKX
|
7.2 | Kd | 28 | — | |
NRUVICOXXLOXCB
|
7.2 | IC50 | 13 | Yes | |
MGMNDPRNDCWSMZ
|
7.2 | IC50 | 12 | Yes |