Target Details
| UniProt AC | O94806 |
|---|---|
| Gene Symbol | PRKD3 |
| Protein Name | Serine/threonine-protein kinase D3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00169 (PH) PF00069 (Pkinase) PF25525 (Ubiquitin_PRKD1_N) |
Summary
- Multi-target molecules 354
- Clinical molecules 117
- Avg pChEMBL 6.89
KEGG Pathways (3)
Active Molecules (354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WTXAWDOYPWWUJL
|
10.1 | IC50 | 11 | — | |
SSXCVTWCXHGTLK
|
9.9 | IC50 | 11 | — | |
KTGVSZYYHHRRGW
|
9.8 | IC50 | 11 | — | |
VIESIZQAHOPEBR
|
9.8 | IC50 | 11 | — | |
NVYBXIDWOJVGQI
|
9.8 | IC50 | 11 | — | |
APVOCXHEVZBCGS
|
9.7 | IC50 | 11 | — | |
DHTLXMRCLSUJPP
|
9.7 | IC50 | 11 | — | |
VVRRZOFLLJAMIK
|
9.4 | IC50 | 11 | — | |
NCAVLXJPDIQUIS
|
9.0 | IC50 | 3 | — | |
XBDRAUPLGHAFCU
|
8.8 | IC50 | 3 | — | |
NVSJOASGKCGXBZ
|
8.8 | IC50 | 16 | Yes | |
QYBVZIIWBRIXMX
|
8.7 | IC50 | 12 | Yes | |
SCJXQZZYGYLKJG
|
8.7 | IC50 | 3 | — | |
OAVGBZOFDPFGPJ
|
8.7 | IC50 | 42 | Yes | |
JZLFYMHIISZQCZ
|
8.7 | IC50 | 12 | Yes | |
AQSSMEORRLJZLU
|
8.5 | Kd | 34 | Yes | |
CHTMRWQLNNRRFJ
|
8.4 | Ki | 70 | — | |
NJPWCTYVEJIQBM
|
8.4 | Ki | 72 | — | |
NLUPJKQOKWBWFC
|
8.4 | Ki | 69 | — | |
RJZDECGDCKOHBV
|
8.4 | Ki | 70 | — | |
KHGPYYFCIAISBU
|
8.3 | Ki | 31 | — | |
WDARYLSSWBWVCU
|
8.3 | Ki | 49 | — | |
YWTBGJGMTBHQTM
|
8.3 | Ki | 65 | — | |
ZGGIYFOLDBTZIL
|
8.3 | Ki | 27 | — | |
XYUFCXJZFZPEJD
|
8.3 | Ki | 23 | Yes | |
BQJRUJTZSGYBEZ
|
8.2 | Kd | 13 | Yes | |
SCJXQZZYGYLKJG
|
8.2 | IC50 | 3 | — | |
ADMFLILDQJSEIK
|
8.2 | Ki | 72 | — | |
BSFNGHCTZDCQBF
|
8.2 | Ki | 93 | — | |
SAYMBMAHSBYKKR
|
8.2 | IC50 | 12 | Yes | |
HKSZLNNOFSGOKW
|
8.2 | IC50 | 408 | — | |
ZKLJKKASNXVQBZ
|
8.1 | Ki | 27 | — | |
POTTVLREWUNNRO
|
8.1 | IC50 | 17 | Yes | |
UIARLYUEJFELEN
|
8.1 | Kd | 289 | Yes | |
CDXNZQYZADSNCP
|
8.0 | IC50 | 12 | Yes | |
DSXXEELGXBCYNQ
|
8.0 | IC50 | 28 | Yes | |
FFKRSNGYONHGEV
|
8.0 | IC50 | 12 | Yes | |
LPILBMJJRGTKOQ
|
8.0 | Ki | 27 | — | |
OPQUGNXQOSDRMT
|
8.0 | IC50 | 12 | Yes | |
PGWBJRRPIUVOAD
|
8.0 | IC50 | 12 | Yes | |
PUYIXDDMOUMMRR
|
8.0 | Ki | 27 | — | |
VLEFVPMCVJDTHZ
|
8.0 | Ki | 13 | — | |
XNWKXXIGSPPPBH
|
7.9 | Ki | 31 | — | |
PBCZSGKMGDDXIJ
|
7.9 | IC50 | 14 | Yes | |
GPGZMTPPOHCJRE
|
7.8 | IC50 | 16 | Yes | |
SMZYTCQRZVNFFJ
|
7.8 | IC50 | 16 | Yes | |
CXSQMXRQOZZFLD
|
7.8 | IC50 | 18 | — | |
FUMCKNCUEAQHCV
|
7.8 | Ki | 103 | — | |
GCBJDOWIQHMCMR
|
7.8 | Ki | 84 | — | |
NWMPVMMGSHXANZ
|
7.8 | Ki | 58 | — |