Target Details
| UniProt AC | O94804 |
|---|---|
| Gene Symbol | STK10 |
| Protein Name | Serine/threonine-protein kinase 10 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF12474 (PKK) |
Summary
- Multi-target molecules 106
- Clinical molecules 28
- Avg pChEMBL 6.94
KEGG Pathways (1)
Active Molecules (106)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
10.4 | Kd | 408 | — | |
CXQHYVUVSFXTMY
|
9.3 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
9.3 | Kd | 149 | — | |
ODPGGGTTYSGTGO
|
9.0 | Kd | 153 | — | |
PBCZSGKMGDDXIJ
|
8.5 | Kd | 68 | Yes | |
UIARLYUEJFELEN
|
8.2 | Kd | 289 | Yes | |
MPASHPJAIUOWCK
|
8.2 | Kd | 9 | — | |
VTWWRKFUHCSCEW
|
8.0 | Kd | 19 | — | |
IKENQUDOTQBCJH
|
8.0 | Kd | 18 | — | |
IUGBGEUCXVKGQK
|
8.0 | Kd | 13 | — | |
MVCOAUNKQVWQHZ
|
7.9 | Kd | 54 | Yes | |
JWNPDZNEKVCWMY
|
7.9 | Kd | 57 | Yes | |
YYLKKYCXAOBSRM
|
7.9 | Kd | 191 | — | |
DKZYXHCYPUVGAF
|
7.8 | Kd | 112 | — | |
WINHZLLDWRZWRT
|
7.7 | Kd | 201 | Yes | |
SHPFDGWALWEPGS
|
7.7 | Kd | 35 | — | |
XXJWYDDUDKYVKI
|
7.6 | Kd | 52 | — | |
DQYDZCRLDYVZKY
|
7.6 | IC50 | 5 | — | |
CRZIGHVWJFDSFR
|
7.6 | IC50 | 5 | — | |
MWKSRKSEWLRPBL
|
7.5 | Kd | 1075 | — | |
KTEIFNKAUNYNJU
|
7.4 | Kd | 114 | — | |
NYZXUVGUIAUXBT
|
7.3 | IC50 | 2 | — | |
AFLQKPBFQDXTFP
|
7.3 | Ki | 2 | — | |
WVXNSAVVKYZVOE
|
7.3 | IC50 | 92 | — | |
UBPYILGKFZZVDX
|
7.3 | Kd | 130 | Yes | |
QVOGVAVHOLLLAZ
|
7.2 | Kd | 4 | — | |
YABJJWZLRMPFSI
|
7.2 | Kd | 34 | — | |
NHHQJBCNYHBUSI
|
7.2 | Kd | 220 | — | |
ZHJGWYRLJUCMRT
|
7.2 | Kd | 18 | — | |
ASUGUQWIHMTFJL
|
7.2 | Kd | 18 | — | |
IDPHPRPMCOPJNX
|
7.1 | Ki | 4 | — | |
CLBAMRRPLGIROG
|
7.1 | Ki | 2 | — | |
MFAQYJIYDMLAIM
|
7.1 | Kd | 130 | Yes | |
PJQXOWLFWLVNJN
|
7.1 | IC50 | 2 | — | |
LOLPPWBBNUVNQZ
|
7.1 | Kd | 97 | Yes | |
QQWUGDVOUVUTOY
|
7.1 | Kd | 231 | Yes | |
UHTHHESEBZOYNR
|
7.1 | Kd | 66 | Yes | |
AAKJLRGGTJKAMG
|
7.1 | Kd | 50 | Yes | |
CUIHSIWYWATEQL
|
7.1 | Kd | 61 | Yes | |
CUTWEHCUKIGMHI
|
7.1 | Ki | 2 | — | |
LZYFXQSDTZSWLB
|
7.1 | Ki | 2 | — | |
XZXHXSATPCNXJR
|
7.1 | Kd | 165 | Yes | |
MUOKSQABCJCOPU
|
7.0 | Kd | 36 | — | |
DSXXEELGXBCYNQ
|
7.0 | IC50 | 28 | Yes | |
FYXCQTJVPMWKNZ
|
7.0 | Ki | 2 | — | |
JVTLNYITMMFMKI
|
7.0 | Ki | 2 | — | |
KDKUVYLMPJIGKA
|
7.0 | Kd | 91 | Yes | |
KPRVTRYCSICYGC
|
7.0 | Ki | 2 | — | |
BESNKWPMIMICNM
|
6.9 | Ki | 2 | — | |
GCIKSSRWRFVXBI
|
6.9 | Kd | 109 | Yes |