Target Details
| UniProt AC | O94782 |
|---|---|
| Gene Symbol | USP1 |
| Protein Name | Ubiquitin carboxyl-terminal hydrolase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00443 (UCH) |
Summary
- Multi-target molecules 83
- Clinical molecules 0
- Avg pChEMBL 6.87
KEGG Pathways (1)
Active Molecules (83)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LYHJNDYWNOAVHB
|
8.2 | IC50 | 2 | — | |
PZIQRTRBAXBGJR
|
8.1 | IC50 | 2 | — | |
NMVACJWIYBGMGN
|
8.0 | IC50 | 2 | — | |
DKTUTBQEFKQWJI
|
7.9 | IC50 | 2 | — | |
ZHLIKWVEMREQBZ
|
7.8 | IC50 | 2 | — | |
FMQIYLHZECZAPT
|
7.7 | IC50 | 2 | — | |
BLJFHWMAIJGAAX
|
7.6 | IC50 | 2 | — | |
CKWBMDPUPBWUGR
|
7.6 | IC50 | 2 | — | |
JACYUDVUPWGGPQ
|
7.5 | IC50 | 2 | — | |
VGAZPJKGOOKEAC
|
7.5 | IC50 | 2 | — | |
KCBWAFJCKVKYHO
|
7.5 | IC50 | 2 | — | |
QVMLBEDORILBMR
|
7.4 | IC50 | 2 | — | |
HHMGGJHFUODDEW
|
7.4 | IC50 | 2 | — | |
OKTDDNGPJVMMAE
|
7.4 | IC50 | 2 | — | |
KREXNTZCOVZMKX
|
7.3 | IC50 | 2 | — | |
AAAQFGUYHFJNHI
|
7.3 | IC50 | 252 | — | |
QLICYNOLYRGEQS
|
7.2 | IC50 | 2 | — | |
FSNHHVDTKUQAHF
|
7.2 | IC50 | 2 | — | |
IUSIQRUSYSTHCC
|
7.2 | IC50 | 2 | — | |
XCXCGYSVONOGSX
|
7.2 | IC50 | 2 | — | |
NEFBWAXVDZOLKA
|
7.2 | IC50 | 2 | — | |
QZKHOMCEQNDZDU
|
7.2 | IC50 | 2 | — | |
VUIRVWPJNKZOSS
|
7.1 | IC50 | 3 | — | |
CTWJXIOHGJUZQD
|
7.1 | IC50 | 2 | — | |
AUSSDHANKWMPME
|
7.1 | IC50 | 2 | — | |
VSEXWFQETXEBSQ
|
7.1 | IC50 | 2 | — | |
JMABKMRDRXPQFY
|
7.0 | IC50 | 2 | — | |
VUIRVWPJNKZOSS
|
7.0 | IC50 | 2 | — | |
BCGFWIIBNQKEOS
|
7.0 | IC50 | 2 | — | |
NNCIGEGVIIXSMD
|
7.0 | IC50 | 2 | — | |
WJOIKYCRIINXLC
|
7.0 | IC50 | 2 | — | |
CGSMWZPSTDEJQI
|
6.9 | IC50 | 2 | — | |
CSOBQKMAXFQFRJ
|
6.9 | IC50 | 2 | — | |
LLCXQBXMQPAQFY
|
6.9 | IC50 | 2 | — | |
OHRMASGYMKXPKD
|
6.9 | IC50 | 2 | — | |
VUIRVWPJNKZOSS
|
6.9 | IC50 | 2 | — | |
YPOLYEAWIMDJKF
|
6.9 | IC50 | 2 | — | |
HEBLAQPNWCDYJV
|
6.8 | IC50 | 2 | — | |
UMSWHQPCXIHXOM
|
6.8 | IC50 | 2 | — | |
VUIRVWPJNKZOSS
|
6.8 | IC50 | 2 | — | |
ZNJXHHPWNNHGRG
|
6.8 | IC50 | 2 | — | |
HDAUDUGYMYCFAO
|
6.8 | IC50 | 2 | — | |
IUFMEYGFNRLJAP
|
6.8 | IC50 | 2 | — | |
NSGRWBBLHJWXQZ
|
6.8 | IC50 | 2 | — | |
RFUYFRZYMMYGEE
|
6.8 | IC50 | 2 | — | |
MYVXJHJCBXQWBE
|
6.8 | IC50 | 2 | — | |
MNNNIKGTZLITAR
|
6.8 | IC50 | 2 | — | |
YTFBNZNGGYGAQN
|
6.8 | IC50 | 2 | — | |
ZUGPAPZFXDQYJW
|
6.8 | IC50 | 2 | — | |
IPNIYJAIHGHHOQ
|
6.7 | IC50 | 2 | — |