Target Details
| UniProt AC | O94768 |
|---|---|
| Gene Symbol | STK17B |
| Protein Name | Serine/threonine-protein kinase 17B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 68
- Clinical molecules 8
- Avg pChEMBL 6.98
Active Molecules (68)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QSDUMEKQISKWQM
|
9.1 | IC50 | 2 | — | |
YYLKKYCXAOBSRM
|
8.3 | Kd | 191 | — | |
UIARLYUEJFELEN
|
8.3 | Kd | 289 | Yes | |
YQMFNWQNASFQAE
|
8.1 | IC50 | 5 | — | |
HHFBDROWDBDFBR
|
8.1 | Kd | 40 | Yes | |
NHHQJBCNYHBUSI
|
8.0 | Kd | 220 | — | |
XKQNBVAZAFAZFL
|
8.0 | IC50 | 6 | — | |
ZUKXESAZGMJHLJ
|
8.0 | IC50 | 4 | — | |
MAUXTEABCSHUTA
|
8.0 | Kd | 2 | — | |
FNCKZBZRSNSOLA
|
7.8 | IC50 | 2 | — | |
LIMMMAWLSIHXGX
|
7.8 | IC50 | 5 | — | |
VVFCWFGNLTVHBL
|
7.8 | IC50 | 5 | — | |
KJCQGDBVLKOAHP
|
7.7 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.7 | Kd | 213 | — | |
QVJYGMLAIWRCFT
|
7.7 | IC50 | 5 | — | |
HKSZLNNOFSGOKW
|
7.6 | Kd | 408 | — | |
NHXNHCQTGVIMIV
|
7.6 | IC50 | 2 | — | |
HHLFERIUOTYKKU
|
7.6 | Kd | 2 | — | |
MJWLCXWVFUXXNZ
|
7.5 | IC50 | 3 | — | |
IWDISKBCTNXZQH
|
7.5 | Kd | 3 | — | |
QVADIDYLQUXJQI
|
7.5 | Kd | 2 | — | |
BNYXRPMABDQJJR
|
7.5 | IC50 | 5 | — | |
CTMGXPGMEMDNLR
|
7.4 | IC50 | 2 | — | |
JOOXLOJCABQBSG
|
7.3 | Kd | 139 | — | |
HRSFSLVREYGRTM
|
7.1 | IC50 | 2 | — | |
GOYAADNAKVCRJS
|
7.0 | IC50 | 2 | — | |
WINHZLLDWRZWRT
|
7.0 | Kd | 201 | Yes | |
CZBQLMXEBSGXMK
|
6.9 | IC50 | 2 | — | |
FKTPDWVDAWOMKC
|
6.9 | IC50 | 2 | — | |
DPMDOFDIFNBKGS
|
6.8 | IC50 | 2 | — | |
PKEYNQACQWYICF
|
6.8 | IC50 | 6 | — | |
MJPLWOKXLCUJOE
|
6.7 | IC50 | 2 | — | |
RXEFTAHHUZTOCL
|
6.7 | IC50 | 2 | — | |
UUSZNXFMBUWTTJ
|
6.7 | IC50 | 2 | — | |
JGIGRRQUXCRVAK
|
6.7 | IC50 | 2 | — | |
RSZNIJJWHYKJKS
|
6.7 | IC50 | 2 | — | |
GBHDESSDDILIEU
|
6.7 | IC50 | 2 | — | |
GGNAPCQTOZTGTK
|
6.7 | IC50 | 2 | — | |
LPTRUOTUVXADBL
|
6.7 | IC50 | 2 | — | |
OFYQAVFEGWZUOW
|
6.7 | IC50 | 2 | — | |
UOUMREPCEXJVFD
|
6.6 | IC50 | 2 | — | |
SOJKVKSSTDCNFB
|
6.6 | IC50 | 2 | — | |
SQVBZWHGFBQRIR
|
6.6 | IC50 | 5 | Yes | |
VKWOSNVEELXNQZ
|
6.6 | IC50 | 3 | — | |
GTVLFJMUKIZPEJ
|
6.5 | IC50 | 2 | — | |
ZDXPORXWNAYWMZ
|
6.5 | IC50 | 2 | — | |
OJBZKMRHGQTLHT
|
6.5 | IC50 | 2 | — | |
CTNPALGJUAXMMC
|
6.5 | Kd | 151 | — | |
PKYSCANLQNSBRH
|
6.5 | IC50 | 2 | — | |
IODFDZLIZNZVAP
|
6.5 | IC50 | 2 | — |