Target Details
| UniProt AC | O94759 |
|---|---|
| Gene Symbol | TRPM2 |
| Protein Name | Transient receptor potential cation channel subfamily M member 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF18139 (LSDAT_euk) PF25969 (NUDT9_N) PF25508 (TRPM2) |
Summary
- Multi-target molecules 3
- Clinical molecules 0
- Avg pChEMBL 6.83
KEGG Pathways (2)
Active Molecules (3)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UYJZZVDLGDDTCL
|
7.6 | IC50 | 8 | — | |
ADWFEADZGIHPDE
|
6.7 | IC50 | 2 | — | |
RVOUDNBEIXGHJY
|
6.2 | IC50 | 2 | — |