Target Details
| UniProt AC | O76083 |
|---|---|
| Gene Symbol | PDE9A |
| Protein Name | High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00233 (PDEase_I) |
Summary
- Multi-target molecules 62
- Clinical molecules 0
- Avg pChEMBL 7.95
KEGG Pathways (2)
Active Molecules (62)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YEXTUBISPSAGMY
|
7.0 | IC50 | 2 | — | |
BWAOKFFQWLQKFA
|
7.0 | IC50 | 3 | — | |
UWLURVWZRQXQEM
|
7.0 | IC50 | 3 | — | |
GXWSVMJGLJNVHK
|
7.0 | IC50 | 2 | — | |
QHMBSVQNZZTUGM
|
7.0 | IC50 | 13 | — | |
OFZGCAMFVYIIHV
|
6.5 | IC50 | 24 | — | |
CNSTWFCIWOBGDU
|
6.5 | IC50 | 6 | — | |
GDQXJMLXEYSICD
|
6.5 | IC50 | 6 | — | |
MMFHEXODWCOMFW
|
6.3 | IC50 | 3 | — | |
SECKRCOLJRRGGV
|
6.3 | IC50 | 16 | — | |
IKXUQDQGFGOUFF
|
6.0 | IC50 | 2 | — | |
JITUOVWOCIXEEZ
|
6.0 | IC50 | 23 | — |